Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50013236
TargetProlyl hydroxylase EGLN2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 1nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD1 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 1nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563887(CHEMBL4785918)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563885(CHEMBL4796629)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563884(CHEMBL4781541)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563881(CHEMBL4793403)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563886(CHEMBL4799940)
Affinity DataIC50: 2nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563869(CHEMBL4798217)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563888(CHEMBL4782037)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563877(CHEMBL4778991)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563868(CHEMBL4788580)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563879(CHEMBL4796462)
Affinity DataIC50: 5nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563878(CHEMBL4780656)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563873(CHEMBL4791127)
Affinity DataIC50: 6nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563880(CHEMBL4783361)
Affinity DataIC50: 8.10nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563882(CHEMBL4782641)
Affinity DataIC50: 10nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563875(CHEMBL4789540)
Affinity DataIC50: 12nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 14nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD3 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563866(CHEMBL4777567)
Affinity DataIC50: 16nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563865(CHEMBL4780077)
Affinity DataIC50: 24nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563871(CHEMBL4800385)
Affinity DataIC50: 28nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50431015(CHEMBL2338329 | US9115085, Compound A Form A | US9...)
Affinity DataIC50: 32nMAssay Description:Inhibition of HIF-PHD2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563890(CHEMBL4794308)
Affinity DataIC50: 110nMAssay Description:Inhibition of HIF-PHD2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563876(CHEMBL4784668)
Affinity DataIC50: 150nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563867(CHEMBL4786322)
Affinity DataIC50: 210nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563874(CHEMBL4792941)
Affinity DataIC50: 390nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563870(CHEMBL4798994)
Affinity DataIC50: 730nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563887(CHEMBL4785918)
Affinity DataIC50: 900nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 2C8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 1.60E+3nMAssay Description:Reversible inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563872(CHEMBL4788451)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEgl nine homolog 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563883(CHEMBL4796588)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563890(CHEMBL4794308)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563888(CHEMBL4782037)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 3A4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 2B6(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of CYP2B6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 2C19(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 2D6(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50563889(CHEMBL4783524)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed