Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50048098
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50095469([5-(1-Benzyl-1H-indazol-3-yl)-furan-2-yl]-methanol...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204471(CHEMBL3927498)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204481(CHEMBL3899458)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204482(CHEMBL3918550)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204459(CHEMBL3936460)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204484(CHEMBL3908512)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204489(CHEMBL3918157)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204472(CHEMBL3915177)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204473(CHEMBL3946046)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204477(CHEMBL3892315)
Affinity DataIC50: 5.60E+4nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204494(CHEMBL3918408)
Affinity DataIC50: 6.10E+4nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204470(CHEMBL3961295)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204474(CHEMBL3940432)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed