Compile Data Set for Download or QSAR
Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 50047970
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199118(CHEMBL3894825)
Affinity DataIC50: 2nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 5nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 14nMAssay Description:Inhibition of HDAC3 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataIC50: 21nMAssay Description:Displacement of [18F]-FDHT from androgen receptor in human LNCAP/AR cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 23nMAssay Description:Inhibition of HDAC1 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 24nMAssay Description:Inhibition of HDAC2 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199116(CHEMBL3948543)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199115(CHEMBL3921621)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199111(CHEMBL3979648)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199117(CHEMBL3983635)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199122(CHEMBL3926959)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199117(CHEMBL3983635)
Affinity DataIC50: 36nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199118(CHEMBL3894825)
Affinity DataIC50: 43nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199121(CHEMBL3908221)
Affinity DataIC50: 68nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199114(CHEMBL3966165)
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199123(CHEMBL3903756)
Affinity DataIC50: 110nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199111(CHEMBL3979648)
Affinity DataIC50: 170nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199119(CHEMBL3948452)
Affinity DataIC50: 230nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199112(CHEMBL3912767)
Affinity DataIC50: 250nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199116(CHEMBL3948543)
Affinity DataIC50: 280nMAssay Description:Inhibition of HDAC3 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199113(CHEMBL3955013)
Affinity DataIC50: 330nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199124(CHEMBL3974665)
Affinity DataIC50: 350nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199114(CHEMBL3966165)
Affinity DataIC50: 495nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199120(CHEMBL3982650)
Affinity DataIC50: 560nMAssay Description:Displacement of [3H]mibolerone from androgen receptor (unknown origin) in membranes after 24 hrs by HAP adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199118(CHEMBL3894825)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199123(CHEMBL3903756)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199117(CHEMBL3983635)
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of HDAC3 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199118(CHEMBL3894825)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HDAC3 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199122(CHEMBL3926959)
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199117(CHEMBL3983635)
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199117(CHEMBL3983635)
Affinity DataIC50: 2.89E+3nMAssay Description:Inhibition of HDAC1 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199118(CHEMBL3894825)
Affinity DataIC50: 3.15E+3nMAssay Description:Inhibition of HDAC1 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199115(CHEMBL3921621)
Affinity DataIC50: 3.33E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199116(CHEMBL3948543)
Affinity DataIC50: 3.37E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199113(CHEMBL3955013)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of HDAC3 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199113(CHEMBL3955013)
Affinity DataIC50: 6.19E+3nMAssay Description:Inhibition of HDAC1 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199115(CHEMBL3921621)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HDAC3 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199115(CHEMBL3921621)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199121(CHEMBL3908221)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199121(CHEMBL3908221)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HDAC3 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199121(CHEMBL3908221)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HDAC2 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199116(CHEMBL3948543)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199121(CHEMBL3908221)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HDAC1 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199116(CHEMBL3948543)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HDAC1 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199115(CHEMBL3921621)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HDAC1 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199111(CHEMBL3979648)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of HDAC3 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199120(CHEMBL3982650)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of HDAC6 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199113(CHEMBL3955013)
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibition of HDAC2 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199111(CHEMBL3979648)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HDAC2 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50199119(CHEMBL3948452)
Affinity DataIC50: 2.02E+4nMAssay Description:Inhibition of HDAC3 (unknown origin) assessed as inhibition of fluorogenic peptide deacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2018
Entry Details Article
PubMed
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