Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50048179
TargetGlucose-dependent insulinotropic receptor(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207277(CHEMBL3976778)
Affinity DataEC50:  950nMAssay Description:Agonist activity at CREB-LBD and GAL4-DBD fused human GPR119 expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207292(CHEMBL3911786)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at CREB-LBD and GAL4-DBD fused human GPR119 expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50244791((2-Fluoro-4-methanesulfonyl-phenyl)-{6-[4-(3-isopr...)
Affinity DataEC50:  700nMAssay Description:Agonist activity at CREB-LBD and GAL4-DBD fused human GPR119 expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 17nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207291(CHEMBL3902771)
Affinity DataIC50: 73nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207295(CHEMBL3984849)
Affinity DataIC50: 120nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207300(CHEMBL3980269)
Affinity DataIC50: 140nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207293(CHEMBL3892718)
Affinity DataIC50: 140nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207277(CHEMBL3976778)
Affinity DataIC50: 220nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207287(CHEMBL3910158)
Affinity DataIC50: 250nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207290(CHEMBL3901674)
Affinity DataIC50: 250nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207283(CHEMBL3897118)
Affinity DataIC50: 260nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207294(CHEMBL3968249)
Affinity DataIC50: 280nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207278(CHEMBL3898220)
Affinity DataIC50: 300nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207281(CHEMBL3896047)
Affinity DataIC50: 360nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207279(CHEMBL3979866)
Affinity DataIC50: 360nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207289(CHEMBL3920718)
Affinity DataIC50: 400nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207286(CHEMBL3933623)
Affinity DataIC50: 500nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207282(CHEMBL3915044)
Affinity DataIC50: 510nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207285(CHEMBL3972227)
Affinity DataIC50: 610nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207296(CHEMBL3929627)
Affinity DataIC50: 760nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207299(CHEMBL3924059)
Affinity DataIC50: 770nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207280(CHEMBL3945617)
Affinity DataIC50: 800nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207298(CHEMBL3899590)
Affinity DataIC50: 890nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207297(CHEMBL3973741)
Affinity DataIC50: 950nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207284(CHEMBL3927979)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207292(CHEMBL3911786)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50207288(CHEMBL3909049)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed