Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50010033
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534481(CHEMBL4516360)
Affinity DataEC50:  104nMAssay Description:Agonist activity at human CB1R expressed in CHO cells by Ca2+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50068666(4-(2-{3-[1-Naphthalen-1-yl-meth-(E)-ylidene]-3H-in...)
Affinity DataEC50:  257nMAssay Description:Agonist activity at human CB1R expressed in CHO cells by Ca2+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534464(CHEMBL4483714)
Affinity DataEC50:  163nMAssay Description:Agonist activity at human CB2R expressed in CHO cells by Ca2+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534476(CHEMBL4443660)
Affinity DataEC50:  182nMAssay Description:Agonist activity at human CB1R expressed in CHO cells by Ca2+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50068666(4-(2-{3-[1-Naphthalen-1-yl-meth-(E)-ylidene]-3H-in...)
Affinity DataEC50:  138nMAssay Description:Agonist activity at human CB2R expressed in CHO cells by Ca2+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534463(CHEMBL4550629)
Affinity DataEC50:  594nMAssay Description:Agonist activity at human CB2R expressed in CHO cells by Ca2+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50212395(CHEMBL123515)
Affinity DataEC50:  196nMAssay Description:Agonist activity at human CB1R expressed in CHO cells by Ca2+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534464(CHEMBL4483714)
Affinity DataEC50:  141nMAssay Description:Agonist activity at human CB1R expressed in CHO cells by Ca2+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50212395(CHEMBL123515)
Affinity DataEC50:  194nMAssay Description:Agonist activity at human CB2R expressed in CHO cells by Ca2+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534476(CHEMBL4443660)
Affinity DataEC50:  94nMAssay Description:Agonist activity at human CB2R expressed in CHO cells by Ca2+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534464(CHEMBL4483714)
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534464(CHEMBL4483714)
Affinity DataKi:  0.859nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534476(CHEMBL4443660)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534476(CHEMBL4443660)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534485(CHEMBL4435655)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50212395(CHEMBL123515)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534457(CHEMBL4444832)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534481(CHEMBL4516360)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50068669(4-(2-{2-Methyl-3-[1-naphthalen-1-yl-meth-(Z)-ylide...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534481(CHEMBL4516360)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50212395(CHEMBL123515)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534463(CHEMBL4550629)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50353747(JWH-018 | CHEMBL561013)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534498(CHEMBL4474739)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50068666(4-(2-{3-[1-Naphthalen-1-yl-meth-(E)-ylidene]-3H-in...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50068666(4-(2-{3-[1-Naphthalen-1-yl-meth-(E)-ylidene]-3H-in...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534467(CHEMBL4549096)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534497(CHEMBL4438072)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534480(CHEMBL4519883)
Affinity DataKi:  9.90nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534463(CHEMBL4550629)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534485(CHEMBL4435655)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534462(CHEMBL4452573)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50032565((4-Methyl-naphthalen-1-yl)-[1-(2-morpholin-4-yl-et...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534482(CHEMBL4469157)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534475(CHEMBL4473031)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534461(CHEMBL4577001)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534497(CHEMBL4438072)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534487(CHEMBL4459965)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534480(CHEMBL4519883)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50009854(CHEMBL13078 | [1-(2-Morpholin-4-yl-ethyl)-1H-indol...)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534494(CHEMBL4574099)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50032599((4-Methoxy-naphthalen-1-yl)-[1-(2-morpholin-4-yl-e...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534458(CHEMBL4475213)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534491(CHEMBL4452886)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534483(CHEMBL4573761)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534466(CHEMBL4476434)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534474(CHEMBL4461845)
Affinity DataKi:  134nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534460(CHEMBL4442680)
Affinity DataKi:  149nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534486(CHEMBL4471974)
Affinity DataKi:  237nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50534478(CHEMBL4560607)
Affinity DataKi:  436nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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