Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50047626
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180193(AZD2624 | AZD-2624)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180171(CHEMBL3813763)
Affinity DataIC50: 3.90nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180169(CHEMBL3814787)
Affinity DataIC50: 5.60nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180174(CHEMBL3813719)
Affinity DataIC50: 6nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50051293(SB-2234 | 3-Hydroxy-2-phenyl-quinoline-4-carboxyli...)
Affinity DataIC50: 8.40nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180170(CHEMBL3815065)
Affinity DataIC50: 24nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180175(CHEMBL3813835)
Affinity DataIC50: 44nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180168(CHEMBL3814967)
Affinity DataIC50: 154nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180172(CHEMBL3813735)
Affinity DataIC50: 245nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180173(CHEMBL3815072)
Affinity DataIC50: 390nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180176(CHEMBL3814793)
Affinity DataIC50: 965nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180184(CHEMBL3813742)
Affinity DataIC50: 1.53E+3nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180166(CHEMBL3814985)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50180167(CHEMBL3815160)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]His3-MePhe7)-NKB from human NK3R expressed in CHO cell membranes by topcounting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2017
Entry Details Article
PubMed