Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50047578
TargetNeuraminidase(Influenza A virus)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176806(CHEMBL3810328)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of Influenza A virus H5N1 neuraminidase preincubated for 10 mins followed by addition of 2'-(4-methylumbelliferyl)-alpha-D-N-acetylneurami...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176807(CHEMBL3808658)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of Influenza A virus H5N1 neuraminidase preincubated for 10 mins followed by addition of 2'-(4-methylumbelliferyl)-alpha-D-N-acetylneurami...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176810(CHEMBL3808427)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176809(CHEMBL3809329)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176812(CHEMBL3809861)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176862(CHEMBL3809053)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176858(CHEMBL3809579)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176857(CHEMBL3809506)
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176814(CHEMBL3810361)
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of Influenza A virus H5N1 neuraminidase preincubated for 10 mins followed by addition of 2'-(4-methylumbelliferyl)-alpha-D-N-acetylneurami...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176863(CHEMBL3809926)
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176806(CHEMBL3810328)
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176859(CHEMBL3809498)
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176807(CHEMBL3808658)
Affinity DataIC50: 2.02E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176860(CHEMBL3809059)
Affinity DataIC50: 3.07E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176856(CHEMBL3810325)
Affinity DataIC50: 3.75E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176814(CHEMBL3810361)
Affinity DataIC50: 4.12E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176804(CHEMBL3808795)
Affinity DataIC50: 4.47E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176813(CHEMBL3809159)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176811(CHEMBL3810058)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176801(CHEMBL3810366)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176805(CHEMBL3810010)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176802(CHEMBL3810109)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176861(CHEMBL3809833)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(SARS-CoV)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50176803(CHEMBL3808558)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SARS coronavirus recombinant 3CL-PRO expressed in Escherichia coli JM109 cells using Dabcyl-KTSAVLQSGFRKME-Edans as fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2017
Entry Details Article
PubMed