Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50047851
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataKi:  0.620nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in CD1 mouse brain membranes after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193284(CHEMBL3978981)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176980(8-chloro-1-(2',4'-dichlorophenyl)-N-homopiperidin-...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  8.18nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193280(CHEMBL3895744)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193277(CHEMBL3984538)
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176976(8-chloro-1-(2',4'-dichlorophenyl)-N-cyclohexyl-1,4...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193278(CHEMBL3889602)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193279(CHEMBL3914728)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193279(CHEMBL3914728)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176989(8-chloro-1-(2',4'-dichlorophenyl)-N-pyrrolidin-1-y...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176976(8-chloro-1-(2',4'-dichlorophenyl)-N-cyclohexyl-1,4...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193278(CHEMBL3889602)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193285(CHEMBL3917142)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193284(CHEMBL3978981)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-CP55,940 from CB2 receptor in CD1 mouse spleen homogenates after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193281(CHEMBL3927357)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193282(CHEMBL3949933)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176980(8-chloro-1-(2',4'-dichlorophenyl)-N-homopiperidin-...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193285(CHEMBL3917142)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193283(CHEMBL3924830)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193282(CHEMBL3949933)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  55.7nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193281(CHEMBL3927357)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193283(CHEMBL3924830)
Affinity DataKi:  169nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50176989(8-chloro-1-(2',4'-dichlorophenyl)-N-pyrrolidin-1-y...)
Affinity DataKi:  182nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193277(CHEMBL3984538)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]-CP55,940 from CB1 receptor in mouse whole brain membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM50193280(CHEMBL3895744)
Affinity DataKi:  325nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  514nMAssay Description:Displacement of [3H]-CP55,940 from CB2 receptor in CD1 mouse spleen homogenates after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Neuroscienze Pharmaness S.C.A R.L.

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor transfected in CHO cell membranes after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2018
Entry Details Article
PubMed