Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50047846
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193122(CHEMBL3899727)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193123(CHEMBL3954358)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193116(CHEMBL3936771)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193115(CHEMBL3945656)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193112(CHEMBL3966536)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193118(CHEMBL3904118)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193114(CHEMBL3958547)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50300690(CHEMBL576982 | N-(5-tert-Butyl-isoxazol-3-yl)-N'-{...)
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193121(CHEMBL3975030)
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193120(CHEMBL3940328)
Affinity DataIC50: 69nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193110(CHEMBL3924345)
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193111(CHEMBL3931041)
Affinity DataIC50: 76nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193113(CHEMBL3905177)
Affinity DataIC50: 118nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193119(CHEMBL3984002)
Affinity DataIC50: 124nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50056801(CHEMBL3326032)
Affinity DataIC50: 156nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193117(CHEMBL3921068)
Affinity DataIC50: 191nMAssay Description:Inhibition of recombinant human FLT3 expressed in insect Sf21 cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193112(CHEMBL3966536)
Affinity DataIC50: 2.88E+3nMAssay Description:Inhibition of recombinant human ABL1 expressed in insect cells preincubated for 15 mins followed by poly(Glu:Tyr) substrate addition for 30 mins in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50193112(CHEMBL3966536)
Affinity DataIC50: 9.75E+3nMAssay Description:Inhibition of human TIE2 preincubated for 15 mins followed by substrate addition measured after 30 mins in presence of [gamma-32P]ATP by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed