Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50047130
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150108(CHEMBL3770617)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149986(CHEMBL3770889)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149988(CHEMBL3770945)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150109(CHEMBL3770355)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150062(CHEMBL3769896)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149985(CHEMBL3769701)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150066(CHEMBL3771319)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149984(CHEMBL3769593)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150111(CHEMBL3771020)
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149983(CHEMBL3769936)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150110(CHEMBL3771098)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150705(CHEMBL3770102)
Affinity DataIC50: 98nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149992(CHEMBL3769897)
Affinity DataIC50: 157nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149990(CHEMBL3770229)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150018(CHEMBL3769551)
Affinity DataIC50: 207nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150019(CHEMBL3769973)
Affinity DataIC50: 227nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50400050(CHEMBL2177757 | US8604016, 1 | US9938267, Cmpd ID ...)
Affinity DataIC50: 371nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149987(CHEMBL3770357)
Affinity DataIC50: 490nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150015(CHEMBL3770218)
Affinity DataIC50: 540nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149982(CHEMBL3769558)
Affinity DataIC50: 720nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149989(CHEMBL3770066)
Affinity DataIC50: 790nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149991(CHEMBL3771046)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150017(CHEMBL3771176)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150067(CHEMBL3771225)
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150658(CHEMBL3769544)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150659(CHEMBL3770563)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150703(CHEMBL3770921)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150660(CHEMBL3769604)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150065(CHEMBL3770713)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150661(CHEMBL3770033)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50150016(CHEMBL3769448)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed