Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 7322
TargetSerum paraoxonase/arylesterase 1(Human)
Ahi Evran University

LigandPNGBDBM50001839(CHEMBL428647 | taxol | PACLITAXEL)
Affinity DataKi:  1.65E+4nM IC50: 4.20E+4nMpH: 10.5Assay Description:Paraoxonase enzyme activity was determined at 25 °C with paraoxon (1 mM) in 50 mM glycine-NaOH (pH 10.5) containing 1 mM CaCl2. The enzyme assay was ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerum paraoxonase/arylesterase 1(Human)
Ahi Evran University

LigandPNGBDBM50127140(4'-Demethylepipodophyllotoxin 9-(4,6-O-(R)-ethylid...)
Affinity DataKi:  1.31E+5nM IC50: 2.26E+5nMpH: 10.5Assay Description:Paraoxonase enzyme activity was determined at 25 °C with paraoxon (1 mM) in 50 mM glycine-NaOH (pH 10.5) containing 1 mM CaCl2. The enzyme assay was ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerum paraoxonase/arylesterase 1(Human)
Ahi Evran University

LigandPNGBDBM36351(CID148124 | Docetaxel)
Affinity DataKi:  2.91E+5nM IC50: 6.65E+5nMpH: 10.5Assay Description:Paraoxonase enzyme activity was determined at 25 °C with paraoxon (1 mM) in 50 mM glycine-NaOH (pH 10.5) containing 1 mM CaCl2. The enzyme assay was ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerum paraoxonase/arylesterase 1(Human)
Ahi Evran University

LigandPNGBDBM189358(N,3-bis(2-chloroethyl)-2-oxo-1,3,2-oxazaphosphinan...)
Affinity DataKi:  8.97E+6nM IC50: 2.33E+7nMpH: 10.5Assay Description:Paraoxonase enzyme activity was determined at 25 °C with paraoxon (1 mM) in 50 mM glycine-NaOH (pH 10.5) containing 1 mM CaCl2. The enzyme assay was ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed