Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50047290
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50158080(CHEMBL3779935)
Affinity DataEC50:  25nMAssay Description:Agonist activity at histidine-tagged ligand binding domain of human RXRalpha expressed in Escherichia coli BL21 (DE3) by luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at Renilla luciferase/GFP2-tagged RXRalpha homodimer (unknown origin) expressed in HEK293T cells by BRET2 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50157943(CHEMBL3780763)
Affinity DataEC50:  20nMAssay Description:Agonist activity at Renilla luciferase/GFP2-tagged RXRalpha homodimer (unknown origin) expressed in HEK293T cells by BRET2 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50157944(CHEMBL3780806)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at Renilla luciferase/GFP2-tagged RXRalpha homodimer (unknown origin) expressed in HEK293T cells by BRET2 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50157942(CHEMBL3781132)
Affinity DataEC50:  6.31nMAssay Description:Agonist activity at Renilla luciferase/GFP2-tagged RXRalpha homodimer (unknown origin) expressed in HEK293T cells by BRET2 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50158083(CHEMBL3780004)
Affinity DataEC50:  50nMAssay Description:Agonist activity at histidine-tagged ligand binding domain of human RXRalpha expressed in Escherichia coli BL21 (DE3) by luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50158082(CHEMBL3781998)
Affinity DataEC50:  50nMAssay Description:Agonist activity at histidine-tagged ligand binding domain of human RXRalpha expressed in Escherichia coli BL21 (DE3) by luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at histidine-tagged ligand binding domain of human RXRalpha expressed in Escherichia coli BL21 (DE3) by luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50157942(CHEMBL3781132)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at histidine-tagged ligand binding domain of human RXRalpha expressed in Escherichia coli BL21 (DE3) by luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50158079(CHEMBL3781771)
Affinity DataEC50:  126nMAssay Description:Agonist activity at histidine-tagged ligand binding domain of human RXRalpha expressed in Escherichia coli BL21 (DE3) by luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50157943(CHEMBL3780763)
Affinity DataEC50:  20nMAssay Description:Agonist activity at histidine-tagged ligand binding domain of human RXRalpha expressed in Escherichia coli BL21 (DE3) by luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed