Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50047249
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156287(CHEMBL3780199)
Affinity DataKi:  60nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM15613(MCL | Aurorix | 4-chloro-N-[2-(morpholin-4-yl)ethy...)
Affinity DataKi:  110nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156288(CHEMBL3780346)
Affinity DataKi:  290nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156284(CHEMBL3780212)
Affinity DataKi:  350nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataKi:  380nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156289(CHEMBL3780057)
Affinity DataKi:  440nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156286(CHEMBL3780858)
Affinity DataKi:  550nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataKi:  710nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156290(CHEMBL3781033)
Affinity DataKi:  2.16E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM15613(MCL | Aurorix | 4-chloro-N-[2-(morpholin-4-yl)ethy...)
Affinity DataKi:  2.24E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156292(CHEMBL3781838)
Affinity DataKi:  2.58E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156292(CHEMBL3781838)
Affinity DataKi:  2.78E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156291(CHEMBL3780319)
Affinity DataKi:  3.87E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156288(CHEMBL3780346)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156285(CHEMBL3781258)
Affinity DataKi:  4.25E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156284(CHEMBL3780212)
Affinity DataKi:  5.02E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156283(CHEMBL3780097)
Affinity DataKi:  9.55E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156286(CHEMBL3780858)
Affinity DataKi:  1.59E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataKi:  1.69E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataKi:  2.15E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156290(CHEMBL3781033)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156291(CHEMBL3780319)
Affinity DataKi:  3.35E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156285(CHEMBL3781258)
Affinity DataKi:  4.11E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156289(CHEMBL3780057)
Affinity DataKi:  2.01E+5nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156283(CHEMBL3780097)
Affinity DataKi:  2.01E+5nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Birla Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50156287(CHEMBL3780199)
Affinity DataKi:  5.90E+6nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed