Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50047199
TargetLysine-specific histone demethylase 1A(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50153586(CHEMBL3775474 | US10053456, 120 | US9718814, 71 | ...)
Affinity DataIC50: 100nMAssay Description:Inhibition of GST-tagged human LSD1 (172 to 833 residues) expressed in Escherichia coli C43(DE3) pLysS using biotinylated histone H3 mono methylated ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50153590(US9487511, 97 | CHEMBL3774809 | US10053456, 97 | U...)
Affinity DataIC50: 100nMAssay Description:Inhibition of GST-tagged human LSD1 (172 to 833 residues) expressed in Escherichia coli C43(DE3) pLysS using biotinylated histone H3 mono methylated ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50153591(US9487511, 99 | CHEMBL3775711 | US10053456, 99 | U...)
Affinity DataIC50: 100nMAssay Description:Inhibition of GST-tagged human LSD1 (172 to 833 residues) expressed in Escherichia coli C43(DE3) pLysS using biotinylated histone H3 mono methylated ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50153593(US9487511, 123 | CHEMBL3775351 | US10053456, 123 |...)
Affinity DataIC50: 100nMAssay Description:Inhibition of GST-tagged human LSD1 (172 to 833 residues) expressed in Escherichia coli C43(DE3) pLysS using biotinylated histone H3 mono methylated ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50153589(US9487511, 95 | CHEMBL3775312 | US10053456, 95 | U...)
Affinity DataIC50: 180nMAssay Description:Inhibition of GST-tagged human LSD1 (172 to 833 residues) expressed in Escherichia coli C43(DE3) pLysS using biotinylated histone H3 mono methylated ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50153592(US9487511, 102 | CHEMBL3774654 | US10053456, 102 |...)
Affinity DataIC50: 210nMAssay Description:Inhibition of GST-tagged human LSD1 (172 to 833 residues) expressed in Escherichia coli C43(DE3) pLysS using biotinylated histone H3 mono methylated ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50153588(US9487511, 84 | CHEMBL3775480 | US10053456, 119 | ...)
Affinity DataIC50: 230nMAssay Description:Inhibition of GST-tagged human LSD1 (172 to 833 residues) expressed in Escherichia coli C43(DE3) pLysS using biotinylated histone H3 mono methylated ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50153587(US9487511, 82 | CHEMBL3775248 | US10053456, 82 | U...)
Affinity DataIC50: 240nMAssay Description:Inhibition of GST-tagged human LSD1 (172 to 833 residues) expressed in Escherichia coli C43(DE3) pLysS using biotinylated histone H3 mono methylated ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed