Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50046852
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50415440(GSK-3787 | CHEMBL598608)
Affinity DataIC50: 1.20nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 24 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50: 29nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 40 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50: 30nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 40 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50134238(CHEMBL3740002)
Affinity DataIC50: 241nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 24 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50415440(GSK-3787 | CHEMBL598608)
Affinity DataIC50: 284nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50: 284nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50: 301nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50: 423nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50134237(CHEMBL3740369)
Affinity DataIC50: 598nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50415440(GSK-3787 | CHEMBL598608)
Affinity DataIC50: 648nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50134237(CHEMBL3740369)
Affinity DataIC50: 907nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50: 949nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50415440(GSK-3787 | CHEMBL598608)
Affinity DataIC50: 1.32E+3nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50134238(CHEMBL3740002)
Affinity DataIC50: 1.43E+3nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50134239(CHEMBL3740264)
Affinity DataIC50: 1.93E+3nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oslo

Curated by ChEMBL
LigandPNGBDBM50134237(CHEMBL3740369)
Affinity DataIC50: 4.22E+3nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed