Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50046993
Affinity DataEC50: 5.10nMAssay Description:Agonist activity at rat mu opioid receptor transfected in C6 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.850nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cell membrane by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Partial agonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced twitchesMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at rat delta opioid receptor transfected in C6 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 73nMAssay Description:Partial agonist activity at mu opioid receptor (unknown origin) expressed in CHO cell membrane assessed as stimulation of [35S]GTP-gamma-S bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at rat delta opioid receptor transfected in C6 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.10nMAssay Description:Agonist activity at rat mu opioid receptor transfected in C6 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0813nMAssay Description:Agonist activity at human delta-opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.80nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Agonist activity at mu opioid receptor (unknown origin) assessed as [35S]GTPgammaS binding by cell based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at delta-opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 36nMAssay Description:Partial agonist activity at delta opioid receptor (unknown origin) assessed as inhibition of adenylyl cyclase activityMore data for this Ligand-Target Pair
Affinity DataEC50: 0.870nMAssay Description:Partial agonist activity at delta opioid receptor (unknown origin) assessed as [35S]GTPgammaS binding by cell based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Agonist activity at delta-opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 4.30nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cell membrane by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0200nMAssay Description:Agonist activity at delta-opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced twitchesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at human delta opioid receptor expressed in CHO cell membrane assessed as inhibition of DAMGO-induced [35S]-GTP-gammaS bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at human delta opioid receptor in CD1 mouse assessed as electrically induced twitchesMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Antagonist activity at human delta opioid receptor expressed in CHO cell membrane assessed as inhibition of DAMGO-induced [35S]-GTP-gammaS bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Binding affinity at mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+3nMAssay Description:Binding affinity at delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Binding affinity at mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0160nMAssay Description:Binding affinity at mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0210nMAssay Description:Binding affinity at delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0310nMAssay Description:Binding affinity at mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0420nMAssay Description:Binding affinity at mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0490nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0490nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0730nMAssay Description:Binding affinity to kappa opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0780nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity at mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.143nMAssay Description:Binding affinity at mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.151nMAssay Description:Displacement of [3H]DPN from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity at delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity at delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Binding affinity to kappa opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]DPDPE from mu opioid receptor in albino Sprague-Dawley rat after 90 mins by liquid scintillationMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.259nMAssay Description:Binding affinity at delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]diprenorphine from rat mu opioid receptor transfected in C6 cells by liquid scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity at mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Binding affinity at delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Displacement of [3H]DAMGO from kappa opioid receptor in albino Sprague-Dawley rat after 90 mins by liquid scintillationMore data for this Ligand-Target Pair
