Compile Data Set for Download or QSAR
Report error Found 89 Enz. Inhib. hit(s) with all data for entry = 50006370
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499239(CHEMBL3734777)
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to human plasma kallikrein by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKd:  737nMAssay Description:Binding affinity to human plasma kallikrein by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKd:  3nMAssay Description:Binding affinity to human plasma kallikrein by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  8nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  9.90nMAssay Description:Inhibition of human wild-type plasma kallikrein catalytic domain after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  14nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  22nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  27nMAssay Description:Inhibition of mouse plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  32nMAssay Description:Inhibition of human plasma kallikrein catalytic domain E217A mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  43nMAssay Description:Inhibition of mouse plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  45nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  50nMAssay Description:Inhibition of mouse plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  54nMAssay Description:Inhibition of human plasma kallikrein catalytic domain G99Y mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499242(CHEMBL3736473)
Affinity DataKi:  64nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  136nMAssay Description:Inhibition of human plasma kallikrein catalytic domain G99Y mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  166nMAssay Description:Inhibition of human plasma kallikrein catalytic domain E217R mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetKallikrein-1(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  201nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetKallikrein-1(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  384nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499239(CHEMBL3734777)
Affinity DataKi:  550nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetKallikrein-1(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  833nMAssay Description:Inhibition of human KLK1 after 15 mins using Val-Leu-Lys-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  907nMAssay Description:Inhibition of human wild-type plasma kallikrein catalytic domain after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  938nMAssay Description:Inhibition of human plasma kallikrein catalytic domain E217A mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  1.58E+3nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  1.69E+3nMAssay Description:Inhibition of human plasma kallikrein catalytic domain E217R mutant after 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  2.56E+3nMAssay Description:Inhibition of human coagulation factor 11a after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasminogen(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  2.97E+3nMAssay Description:Inhibition of mouse plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasminogen(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  3.42E+3nMAssay Description:Inhibition of mouse plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasminogen(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  3.67E+3nMAssay Description:Inhibition of mouse plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  3.97E+3nMAssay Description:Inhibition of human coagulation factor 11a after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  4.61E+3nMAssay Description:Inhibition of mouse plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  6.63E+3nMAssay Description:Inhibition of human coagulation factor 11a after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasminogen(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  9.80E+3nMAssay Description:Inhibition of human plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasminogen(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  1.06E+4nMAssay Description:Inhibition of human plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  1.21E+4nMAssay Description:Inhibition of human coagulation factor 11a after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasminogen(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  1.25E+4nMAssay Description:Inhibition of human plasmin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi:  1.41E+4nMAssay Description:Inhibition of bovine beta-trypsin after 15 mins using Bz-Ile-Glu(g-OR)-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  1.45E+4nMAssay Description:Inhibition of bovine beta-trypsin after 15 mins using Bz-Ile-Glu(g-OR)-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi:  1.82E+4nMAssay Description:Inhibition of bovine beta-trypsin after 15 mins using Bz-Ile-Glu(g-OR)-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499239(CHEMBL3734777)
Affinity DataKi:  2.07E+4nMAssay Description:Inhibition of bovine beta-trypsin after 15 mins using Bz-Ile-Glu(g-OR)-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetSerine protease 1(Bovine)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi:  7.34E+4nMAssay Description:Inhibition of bovine beta-trypsin after 15 mins using Bz-Ile-Glu(g-OR)-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  9.30E+4nMAssay Description:Inhibition of human uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse tPA after 15 mins using Z-D-Arg-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human tPAn after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499239(CHEMBL3734777)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human plasma kallikrein for 15 mins using H-D-Pro-Phe-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human tPAn after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499239(CHEMBL3734777)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human activated protein C after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetProthrombin(Mouse)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse thrombin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetProthrombin(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human thrombin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetProthrombin(Human)
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human thrombin after 15 mins using H-D-Ile-Pro-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
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