Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50046823
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133328(CHEMBL3632807)
Affinity DataIC50: 400nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133350(CHEMBL2036880 | 8-methoxy-beta-lapachone)
Affinity DataIC50: 600nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM81348(R115 (Reactive Blue 2) | β-Lapachone (A3) | b...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133331(CHEMBL3632804)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133340(CHEMBL3635001)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133329(CHEMBL3632806)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133347(CHEMBL3634995)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM81348(R115 (Reactive Blue 2) | β-Lapachone (A3) | b...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133351(CHEMBL177685)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133349(CHEMBL3634993)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133338(CHEMBL3635003)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133336(CHEMBL3632800)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133332(CHEMBL3183233)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133337(CHEMBL3632799)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133339(CHEMBL3635002)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133346(CHEMBL3634996)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133352(CHEMBL3632808)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133330(CHEMBL3632805)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133354(CHEMBL3632809)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133335(CHEMBL3632801)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133333(CHEMBL3632803)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133334(CHEMBL3632802)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133344(CHEMBL3634998)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133343(CHEMBL3634999)
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133342(CHEMBL3635000)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133348(CHEMBL3634994)
Affinity DataIC50: 2.04E+4nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133345(CHEMBL3634997)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Human)
Institute of Basic Science (Ibs)

Curated by ChEMBL
LigandPNGBDBM50133341(CHEMBL1966084)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MALT1 in human Jurkat cell lysate preincubated for 2 hrs followed by addition of 25 uM Ac-LRSR-AMC substrate for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2016
Entry Details Article
PubMed