Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50046843
TargetGlycogen synthase kinase-3 beta(Human)
Angelini

Curated by ChEMBL
LigandPNGBDBM186204(US9163013, 21)
Affinity DataIC50: 9.60nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Angelini

Curated by ChEMBL
LigandPNGBDBM186202(US9163013, 19)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Angelini

Curated by ChEMBL
LigandPNGBDBM186200(US9163013, 17)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Angelini

Curated by ChEMBL
LigandPNGBDBM50134914(CHEMBL3735730)
Affinity DataIC50: 210nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Angelini

Curated by ChEMBL
LigandPNGBDBM50134187(CHEMBL3735506 | US9611249, Compound 8 | US11472795...)
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant ERK5 by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Angelini

Curated by ChEMBL
LigandPNGBDBM186201(US9163013, 18)
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50134187(CHEMBL3735506 | US9611249, Compound 8 | US11472795...)
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant DYRK2 by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Angelini

Curated by ChEMBL
LigandPNGBDBM50134187(CHEMBL3735506 | US9611249, Compound 8 | US11472795...)
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant GRK2 by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Angelini

Curated by ChEMBL
LigandPNGBDBM50134188(CHEMBL3735095)
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed