Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50046809
Target5-hydroxytryptamine receptor 2A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human 5-HT2A receptor assessed as inhibition of 5-HT-mediated internal calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
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PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: <300nMAssay Description:Displacement of [3H]-Pentazocine from recombinant human sigma-1 receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
TargetSodium-dependent dopamine transporter(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: <300nMAssay Description:Displacement of [3H]-WIN35428 from recombinant human DAT after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
TargetAlpha-2A adrenergic receptor(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: <300nMAssay Description:Displacement of [3H]-Clonidine from recombinant human adrenergic alpha2A receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
Target5-hydroxytryptamine receptor 6(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: <300nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
Target5-hydroxytryptamine receptor 2C(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: <300nMAssay Description:Displacement of [3H]-Mesulergine from recombinant human 5-HT2C receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
TargetD(1A) dopamine receptor(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-SCH233930 from recombinant human dopamine D1 receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
TargetTranslocator protein(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-PK11195 from recombinant human PBR after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-Tiotidine from recombinant human muscarinic M5 receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
TargetHistamine H2 receptor(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-Tiotidine from recombinant human histamine H2 receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
TargetD(3) dopamine receptor(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-N-methylspiperone from recombinant human dopamine D3 receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
TargetAlpha-2C adrenergic receptor(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-Clonidine from recombinant human adrenergic alpha2C receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-Clonidine from recombinant human adrenergic alpha2B receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT7 receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
Target5-hydroxytryptamine receptor 3A(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-LY278584 from recombinant human 5-HT3 receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
Target5-hydroxytryptamine receptor 2B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT2B receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
Target5-hydroxytryptamine receptor 1E(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-5-HT from recombinant human 5-HT1E receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
Target5-hydroxytryptamine receptor 1D(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-GR127543 from recombinant human 5-HT1D receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
Target5-hydroxytryptamine receptor 1B(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50132341(CHEMBL3633757)
Affinity DataKi: >900nMAssay Description:Displacement of [3H]-GR127543 from recombinant human 5-HT1B receptor after 1.5 hrs by Microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed