Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 6986
TargetRhomboid protease GlpG(Haemophilus influenzae (g-Proteobacteria))
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 660nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid domain-containing protein(Thermotoga maritima (strain ATCC 43589 / MSB8 / DS...)
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 1.00E+3nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid domain-containing protein(Aquifex aeolicus (strain VF5))
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 1.10E+3nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid domain-containing protein(Aquifex aeolicus (strain VF5))
Technische Universität München

LigandPNGBDBM165194(4‐Chloro‐7‐nitro‐3‐[...)
Affinity DataIC50: 1.70E+3nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid protease GluP [F193S,L370F,L379S,R499W](Bacillus subtilis (strain 168))
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 4.10E+3nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid protease GlpG(Haemophilus influenzae (g-Proteobacteria))
Technische Universität München

LigandPNGBDBM165194(4‐Chloro‐7‐nitro‐3‐[...)
Affinity DataIC50: 4.60E+3nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetAN1-type domain-containing protein(Archaeoglobus fulgidus (AfROM))
Technische Universität München

LigandPNGBDBM165195((4S)‐4‐(pent‐4‐yn‐1&...)
Affinity DataIC50: 5.00E+3nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetAN1-type domain-containing protein(Archaeoglobus fulgidus (AfROM))
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 8.10E+3nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid protease AarA(Providencia stuartii)
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid protease AarA(Providencia stuartii)
Technische Universität München

LigandPNGBDBM165194(4‐Chloro‐7‐nitro‐3‐[...)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid domain-containing protein(Pyrococcus horikoshii (strain ATCC 700860 / DSM 12...)
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 1.60E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 1.90E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid-related protein 3(Mouse)
Technische Universität München

LigandPNGBDBM165194(4‐Chloro‐7‐nitro‐3‐[...)
Affinity DataIC50: 2.40E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid domain-containing protein(Pyrococcus horikoshii (strain ATCC 700860 / DSM 12...)
Technische Universität München

LigandPNGBDBM165194(4‐Chloro‐7‐nitro‐3‐[...)
Affinity DataIC50: 2.50E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid protease GluP [F193S,L370F,L379S,R499W](Bacillus subtilis (strain 168))
Technische Universität München

LigandPNGBDBM165194(4‐Chloro‐7‐nitro‐3‐[...)
Affinity DataIC50: 2.50E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetGlpG protein(Vibrio cholerae)
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 2.70E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid domain-containing protein(Thermotoga maritima (strain ATCC 43589 / MSB8 / DS...)
Technische Universität München

LigandPNGBDBM165196((4S)‐4‐(pent‐4‐yn‐1&...)
Affinity DataIC50: 2.70E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid domain-containing protein(Thermotoga maritima (strain ATCC 43589 / MSB8 / DS...)
Technische Universität München

LigandPNGBDBM165194(4‐Chloro‐7‐nitro‐3‐[...)
Affinity DataIC50: 2.80E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid-related protein 1(Mouse)
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 2.80E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid-related protein 1(Mouse)
Technische Universität München

LigandPNGBDBM165194(4‐Chloro‐7‐nitro‐3‐[...)
Affinity DataIC50: 3.90E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Technische Universität München

LigandPNGBDBM165197((4S)‐3‐butyl‐4‐(pent‐...)
Affinity DataIC50: 4.40E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid domain-containing protein(Thermotoga maritima (strain ATCC 43589 / MSB8 / DS...)
Technische Universität München

LigandPNGBDBM165197((4S)‐3‐butyl‐4‐(pent‐...)
Affinity DataIC50: 4.80E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid protease GlpG(Haemophilus influenzae (g-Proteobacteria))
Technische Universität München

LigandPNGBDBM165195((4S)‐4‐(pent‐4‐yn‐1&...)
Affinity DataIC50: 6.50E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetRhomboid-related protein 3(Mouse)
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 7.00E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed
TargetGlpG protein(Vibrio cholerae)
Technische Universität München

LigandPNGBDBM165194(4‐Chloro‐7‐nitro‐3‐[...)
Affinity DataIC50: 7.60E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2016
Entry Details Article
PubMed