Compile Data Set for Download or QSAR
Report error Found 67 Enz. Inhib. hit(s) with all data for entry = 50046357
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107864(CHEMBL3601192)
Affinity DataIC50: 0.740nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108079(CHEMBL3601079)
Affinity DataIC50: 2nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108087(CHEMBL3601071 | US9598440, 69)
Affinity DataIC50: 3nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107848(CHEMBL3601185)
Affinity DataIC50: 4nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108086(CHEMBL3601072 | US9598440, 66)
Affinity DataIC50: 4nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108080(CHEMBL3601078)
Affinity DataIC50: 6nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108083(CHEMBL3601075)
Affinity DataIC50: 7nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107915(CHEMBL3601189)
Affinity DataIC50: 8nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108084(CHEMBL3601074)
Affinity DataIC50: 11nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107847(CHEMBL3601186)
Affinity DataIC50: 11nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108078(CHEMBL3601080)
Affinity DataIC50: 12nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108085(CHEMBL3601073)
Affinity DataIC50: 12nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108082(CHEMBL3601076)
Affinity DataIC50: 12nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107852(CHEMBL3601196 | US9598440, 154)
Affinity DataIC50: 14nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108077(CHEMBL3601081)
Affinity DataIC50: 18nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107915(CHEMBL3601189)
Affinity DataIC50: 25nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107866(CHEMBL3601070)
Affinity DataIC50: 27nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107893(CHEMBL3601190)
Affinity DataIC50: 44nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107864(CHEMBL3601192)
Affinity DataIC50: 55nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107848(CHEMBL3601185)
Affinity DataIC50: 87nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108012(CHEMBL3601187)
Affinity DataIC50: 89nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107847(CHEMBL3601186)
Affinity DataIC50: 94nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108011(CHEMBL3601188)
Affinity DataIC50: 94nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107862(CHEMBL3601193 | US9598440, 152)
Affinity DataIC50: 113nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107865(CHEMBL3601191)
Affinity DataIC50: 155nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107855(CHEMBL3601194 | US9598440, 153)
Affinity DataIC50: 204nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107866(CHEMBL3601070)
Affinity DataIC50: 216nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107893(CHEMBL3601190)
Affinity DataIC50: 341nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107851(CHEMBL3601197 | US9598440, 155)
Affinity DataIC50: 373nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108081(CHEMBL3601077)
Affinity DataIC50: 647nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108016(CHEMBL3601083 | US9598440, 41)
Affinity DataIC50: 852nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108014(CHEMBL3601085)
Affinity DataIC50: 932nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107854(CHEMBL3601195 | US9598440, 151)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108015(CHEMBL3601084 | US9598440, 40)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107852(CHEMBL3601196 | US9598440, 154)
Affinity DataIC50: 3.45E+3nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108013(CHEMBL3601086)
Affinity DataIC50: 6.01E+3nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107850(CHEMBL3601198 | US9598440, 158)
Affinity DataIC50: 9.51E+3nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107849(CHEMBL3601199 | US9598440, 157)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108017(CHEMBL3601082)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107866(CHEMBL3601070)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107852(CHEMBL3601196 | US9598440, 154)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107864(CHEMBL3601192)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107915(CHEMBL3601189)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107847(CHEMBL3601186)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107848(CHEMBL3601185)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107893(CHEMBL3601190)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107852(CHEMBL3601196 | US9598440, 154)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107864(CHEMBL3601192)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107866(CHEMBL3601070)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 2C9(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50107893(CHEMBL3601190)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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