Compile Data Set for Download or QSAR
Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50045963
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089076(CHEMBL3577642)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088858(CHEMBL3577566)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088791(CHEMBL3577634)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089074(CHEMBL3577643)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088791(CHEMBL3577634)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088855(CHEMBL3577632)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088855(CHEMBL3577632)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088858(CHEMBL3577566)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088897(CHEMBL3577644)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088896(CHEMBL3577645)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089083(CHEMBL3577635)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089083(CHEMBL3577635)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089074(CHEMBL3577643)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088857(CHEMBL3577567)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088854(CHEMBL3577633)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088856(CHEMBL3577631)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088854(CHEMBL3577633)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088856(CHEMBL3577631)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088897(CHEMBL3577644)
Affinity DataIC50: 7nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 18nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088859(CHEMBL3577565)
Affinity DataIC50: 20nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089077(CHEMBL3577641)
Affinity DataIC50: 21nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089077(CHEMBL3577641)
Affinity DataIC50: 21nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089082(CHEMBL3577636)
Affinity DataIC50: 23nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089076(CHEMBL3577642)
Affinity DataIC50: 23nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089081(CHEMBL3577637)
Affinity DataIC50: 23nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089082(CHEMBL3577636)
Affinity DataIC50: 23nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089079(CHEMBL3577639)
Affinity DataIC50: 23nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089077(CHEMBL3577641)
Affinity DataIC50: 23nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089074(CHEMBL3577643)
Affinity DataIC50: 24nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088858(CHEMBL3577566)
Affinity DataIC50: 25nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089081(CHEMBL3577637)
Affinity DataIC50: 32nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089078(CHEMBL3577640)
Affinity DataIC50: 34nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088897(CHEMBL3577644)
Affinity DataIC50: 35nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088895(CHEMBL3577563)
Affinity DataIC50: 35nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 37nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089078(CHEMBL3577640)
Affinity DataIC50: 43nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088859(CHEMBL3577565)
Affinity DataIC50: 43nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088894(CHEMBL3577564)
Affinity DataIC50: 43nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089079(CHEMBL3577639)
Affinity DataIC50: 43nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088896(CHEMBL3577645)
Affinity DataIC50: 44nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088894(CHEMBL3577564)
Affinity DataIC50: 44nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088857(CHEMBL3577567)
Affinity DataIC50: 46nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088896(CHEMBL3577645)
Affinity DataIC50: 47nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088857(CHEMBL3577567)
Affinity DataIC50: 54nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088895(CHEMBL3577563)
Affinity DataIC50: 54nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089081(CHEMBL3577637)
Affinity DataIC50: 56nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088856(CHEMBL3577631)
Affinity DataIC50: 57nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088895(CHEMBL3577563)
Affinity DataIC50: 65nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088894(CHEMBL3577564)
Affinity DataIC50: 66nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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