Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50045668
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073602(CHEMBL3408973)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Human)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL63064 | N-(2,5-Dimethoxy-benzyl)-N-(5-fluoro...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073596(CHEMBL3408967)
Affinity DataKi:  0.310nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073597(CHEMBL3408968)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073600(CHEMBL3408971)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50229594(N-(2-methoxybenzyl)-N-(4-phenoxypyridin-3-yl)aceta...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of rat TSPOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073598(CHEMBL3408969)
Affinity DataKi:  0.770nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073591(CHEMBL3408960)
Affinity DataKi:  0.860nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Human)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073588(CHEMBL3408974)
Affinity DataKi:  0.870nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073595(CHEMBL3408966)
Affinity DataKi:  0.990nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073603(CHEMBL3408963)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073599(CHEMBL3408970)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073592(CHEMBL3408961)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073601(CHEMBL3408972)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073604(CHEMBL3408964)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073589(CHEMBL3408958)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073590(CHEMBL3408959)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Human)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50229594(N-(2-methoxybenzyl)-N-(4-phenoxypyridin-3-yl)aceta...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073593(CHEMBL3408962)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  3nMAssay Description:Inhibition of rat TSPOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetTranslocator protein(Rat)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50073594(CHEMBL3408965)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranslocator protein(Human)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed