Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50045494
TargetCannabinoid receptor 1(Mouse)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50065011(CHEMBL3402653)
Affinity DataIC50: 31nMAssay Description:Partial agonist activity at mouse CB1 receptor by vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50399157(CHEMBL2179724)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]HU-243 from CB2 receptor (unknown origin) transfected in human COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Rat)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50399157(CHEMBL2179724)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to rat CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed