Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50045693
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075577(CHEMBL3415556)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of tumorigenic wild type B-Raf in human IPC-298 cells with Ras mutation assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075581(CHEMBL3415555)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of tumorigenic wild type B-Raf in human IPC-298 cells with Ras mutation assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075576(CHEMBL3415554)
Affinity DataEC50: <500nMAssay Description:Activation of tumorigenic wild type B-Raf in human IPC-298 cells with Ras mutation assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075578(CHEMBL3415553)
Affinity DataKd:  130nMAssay Description:Binding affinity to B-Raf V600E mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075576(CHEMBL3415554)
Affinity DataKd:  140nMAssay Description:Binding affinity to B-Raf V600E mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075581(CHEMBL3415555)
Affinity DataKd:  550nMAssay Description:Binding affinity to B-Raf V600E mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075577(CHEMBL3415556)
Affinity DataKd:  1.41E+3nMAssay Description:Binding affinity to B-Raf V600E mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075578(CHEMBL3415553)
Affinity DataKd:  62nMAssay Description:Binding affinity to wild type B-Raf (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075576(CHEMBL3415554)
Affinity DataKd:  100nMAssay Description:Binding affinity to wild type B-Raf (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075581(CHEMBL3415555)
Affinity DataKd:  400nMAssay Description:Binding affinity to wild type B-Raf (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075577(CHEMBL3415556)
Affinity DataKd:  690nMAssay Description:Binding affinity to wild type B-Raf (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075576(CHEMBL3415554)
Affinity DataIC50: 13nMAssay Description:Inhibition of B-Raf V600E mutant (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075578(CHEMBL3415553)
Affinity DataIC50: 31nMAssay Description:Inhibition of B-Raf V600E mutant (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075577(CHEMBL3415556)
Affinity DataIC50: 100nMAssay Description:Inhibition of B-Raf V600E mutant (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075581(CHEMBL3415555)
Affinity DataIC50: 100nMAssay Description:Inhibition of B-Raf V600E mutant (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075578(CHEMBL3415553)
Affinity DataIC50: 100nMAssay Description:Inhibition of wild type B-Raf (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075576(CHEMBL3415554)
Affinity DataIC50: 160nMAssay Description:Inhibition of wild type B-Raf (unknown origin) assessed as inhibition of phosphorylation of peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075576(CHEMBL3415554)
Affinity DataIC50: 800nMAssay Description:Inhibition of B-Raf V600E mutant in human A375 cells assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075581(CHEMBL3415555)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of B-Raf V600E mutant in human A375 cells assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Umr Cnrs-Universit£

Curated by ChEMBL
LigandPNGBDBM50075577(CHEMBL3415556)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of B-Raf V600E mutant in human A375 cells assessed as phosphorylation of ERKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed