Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50006311
TargetREST corepressor 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50464671(CHEMBL3621615)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of recombinant LSD1/CoREST (unknown origin) assessed as residual activity for 30 mins to 4 hrs by fluorescence based assay relative to con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50498660(CHEMBL1605826)
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of recombinant LSD1/CoREST (unknown origin) assessed as residual activity for 30 mins to 4 hrs by fluorescence based assay relative to con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of MAOA (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of MAOB (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataIC50: 2.07E+4nMAssay Description:Inhibition of recombinant LSD1/CoREST (unknown origin) assessed as residual activity for 30 mins to 4 hrs by fluorescence based assay relative to con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50498660(CHEMBL1605826)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MAOB (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50464671(CHEMBL3621615)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MAOA (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50464671(CHEMBL3621615)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MAOB (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50498660(CHEMBL1605826)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MAOA (unknown origin) by luminiscent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50464671(CHEMBL3621615)
Affinity DataKi:  2.20E+3nMAssay Description:Competitive inhibition of LSD1 (unknown origin) incubated for 30 mins using H3K4me2 substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed