Report error Found 109 Enz. Inhib. hit(s) with all data for entry = 50045612
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human recombinant dopmaine D3 receptor expressed in CHOK1 cells assessed as effect on cAMP levelsMore data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:Agonist activity at human recombinant dopmaine D2L receptor expressed in CHOK1 cells assessed as intracellular Ca2+ levels by aequorin based radiomet...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human dopamine D2 receptor expressed in CHOK1 cells assessed as inhibition of apomorphine-induced calcium mobilization by radi...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity against human recombinant alpha1 receptor expressed in CHOK1 cells assessed as reduction in epinephrine-induced increase in intra...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity against human recombinant dopmaine D2L receptor expressed in CHOK1 cells assessed as reduction in apomorphine-induced increase in...More data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Agonist activity at human dopamine D2 receptor expressed in CHOK1 cells assessed as calcium mobilization by radiometric and luminescence plate counti...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Agonist activity at human 5-HT6 receptor expressed in CHOK1 cells assessed as calcium mobilization by radiometric and luminescence plate counting met...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity against human recombinant 5-HT6 receptor expressed in CHOK1 cells assessed as reduction in serotonin-induced increase in intracel...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity against human recombinant 5-HT1A receptor expressed in CHOK1 cells assessed as reduction in serotonin-induced increase in intrace...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity against human recombinant 5-HT2A receptor expressed in CHOK1 cells assessed as reduction in alpha-methylserotonin-induced increas...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity against human recombinant dopmaine D3 receptor expressed in CHOK1 cells assessed as reduction in dopamine-induced cAMP levelsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as reduction in channel current at holding potential of 0 mV by electrophysiological methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as reduction in channel current at holding potential of 0 mV by electrophysiological methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Displacement of [3H]methylspiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Displacement of [3H]methylspiperone from human D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]methylspiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]RX-821002 from human adrenergic alpha2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]LSD from human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]N-methylspiperone from human recombinant dopamine D2 receptor expressed in CHOK1 cells incubated for 60 mins by scintillation cou...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]N-methylspiperone from human recombinant dopamine D2 receptor expressed in CHOK1 cells incubated for 60 mins by scintillation cou...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]N-methylspiperone from human recombinant dopamine D2 receptor expressed in CHOK1 cells incubated for 60 mins by scintillation cou...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]N-methylspiperone from human recombinant dopamine D2 receptor expressed in CHOK1 cells incubated for 60 mins by scintillation cou...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Displacement of [3H]N-methylspiperone from human recombinant dopamine D2 receptor expressed in CHOK1 cells incubated for 60 mins by scintillation cou...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]methylspiperone from human D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]N-methylspiperone from human recombinant dopamine D2 receptor expressed in CHOK1 cells incubated for 60 mins by scintillation cou...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 6.90nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]methylspiperone from human dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 7.60nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 9.90nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]N-methylspiperone from human recombinant dopamine D2 receptor expressed in CHOK1 cells incubated for 60 mins by scintillation cou...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]N-methylspiperone from human recombinant dopamine D2 receptor expressed in CHOK1 cells incubated for 60 mins by scintillation cou...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
