Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50044763
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029022(CHEMBL3339205)
Affinity DataIC50: 900nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029023(CHEMBL3339204)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029020(CHEMBL3339207)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029021(CHEMBL3339206)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029030(CHEMBL3339201)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029024(CHEMBL3339203)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase PKLR(Human)
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029022(CHEMBL3339205)
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of purified human N-terminal His-tagged PK-R by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029025(CHEMBL3339202)
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase PKLR(Human)
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029022(CHEMBL3339205)
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of purified human N-terminal His-tagged PK-L by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029038(CHEMBL3339199)
Affinity DataIC50: 3.28E+4nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029035(CHEMBL3339200)
Affinity DataIC50: 3.86E+4nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029019(CHEMBL3339208)
Affinity DataIC50: 5.02E+4nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase PKM(Human)
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029022(CHEMBL3339205)
Affinity DataIC50: 5.46E+4nMAssay Description:Inhibition of purified human N-terminal His-tagged PK-M2 by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029040(CHEMBL3339198)
Affinity DataIC50: 5.73E+4nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase PKM(Human)
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029022(CHEMBL3339205)
Affinity DataIC50: 9.59E+4nMAssay Description:Inhibition of purified human N-terminal His-tagged PK-M1 by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029016(CHEMBL3339213)
Affinity DataIC50: 1.48E+5nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029018(CHEMBL3339209)
Affinity DataIC50: 2.72E+5nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
University of British Columbia

Curated by ChEMBL
LigandPNGBDBM50029017(CHEMBL3339212)
Affinity DataIC50: 2.94E+5nMAssay Description:Inhibition of purified methicillin-resistant Staphylococcus aureus N-terminal His-tagged pyruvate kinase by LDH-coupled continuous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed