Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50046197
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098808(CHEMBL3334776)
Affinity DataIC50: 69nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50386812(DOV 21947 | DOV-21947 | EB-1010 | AMITIFADINE HYDR...)
Affinity DataIC50: 71nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098901(CHEMBL3334802)
Affinity DataIC50: 136nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098806(CHEMBL3334769)
Affinity DataIC50: 157nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50386812(DOV 21947 | DOV-21947 | EB-1010 | AMITIFADINE HYDR...)
Affinity DataIC50: 159nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098896(CHEMBL3334800)
Affinity DataIC50: 206nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098808(CHEMBL3334776)
Affinity DataIC50: 238nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098893(CHEMBL3334797)
Affinity DataIC50: 247nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098863(CHEMBL3334796)
Affinity DataIC50: 250nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098899(CHEMBL3334773)
Affinity DataIC50: 291nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098806(CHEMBL3334769)
Affinity DataIC50: 325nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098900(CHEMBL3334783)
Affinity DataIC50: 328nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098897(CHEMBL3334801)
Affinity DataIC50: 338nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098896(CHEMBL3334800)
Affinity DataIC50: 357nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098901(CHEMBL3334802)
Affinity DataIC50: 363nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098897(CHEMBL3334801)
Affinity DataIC50: 374nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098893(CHEMBL3334797)
Affinity DataIC50: 379nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098808(CHEMBL3334776)
Affinity DataIC50: 389nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098895(CHEMBL3334799)
Affinity DataIC50: 399nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098810(CHEMBL3334794)
Affinity DataIC50: 401nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50386812(DOV 21947 | DOV-21947 | EB-1010 | AMITIFADINE HYDR...)
Affinity DataIC50: 412nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098863(CHEMBL3334796)
Affinity DataIC50: 425nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098899(CHEMBL3334773)
Affinity DataIC50: 426nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098895(CHEMBL3334799)
Affinity DataIC50: 428nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098809(CHEMBL3334793)
Affinity DataIC50: 449nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098893(CHEMBL3334797)
Affinity DataIC50: 478nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098810(CHEMBL3334794)
Affinity DataIC50: 495nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098896(CHEMBL3334800)
Affinity DataIC50: 501nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098894(CHEMBL3334798)
Affinity DataIC50: 546nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098894(CHEMBL3334798)
Affinity DataIC50: 602nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098806(CHEMBL3334769)
Affinity DataIC50: 621nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098894(CHEMBL3334798)
Affinity DataIC50: 634nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098898(CHEMBL3334772)
Affinity DataIC50: 635nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098902(CHEMBL3334771)
Affinity DataIC50: 852nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098810(CHEMBL3334794)
Affinity DataIC50: 863nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098807(CHEMBL3334770)
Affinity DataIC50: 905nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098863(CHEMBL3334796)
Affinity DataIC50: 986nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098811(CHEMBL3334795)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of [3H]-serotonin uptake in human SERT expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098809(CHEMBL3334793)
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098811(CHEMBL3334795)
Affinity DataIC50: 2.54E+3nMAssay Description:Inhibition of [3H]-NE uptake in human norepinephrine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50098897(CHEMBL3334801)
Affinity DataIC50: 8.19E+3nMAssay Description:Inhibition of [3H]-DA uptake in human dopamine transporter expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed