Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 8810
TargetTransmembrane protease serine 2(Human)
Fred Hutchinson Cancer Research Center

LigandPNGBDBM50239965(CHEBI:77032 | Bromhexine)
Affinity DataIC50: 750nMAssay Description:To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransmembrane protease serine 2(Human)
Fred Hutchinson Cancer Research Center

LigandPNGBDBM420291(0591-5329 | 4-(Methoxycarbonyl)phenyl thiophene-2-...)
Affinity DataIC50: 930nMAssay Description:To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several c...More data for this Ligand-Target Pair
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TargetTransmembrane protease serine 2(Human)
Fred Hutchinson Cancer Research Center

LigandPNGBDBM50022172(CHEMBL275000 | cid_5395514 | (7-Hydroxy-2-oxo-2H-c...)
Affinity DataIC50: 1.37E+3nMAssay Description:To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransmembrane protease serine 2(Human)
Fred Hutchinson Cancer Research Center

LigandPNGBDBM420294(8008-1235 | N-[4-(4-chlorophenyl)-3-ethyl-1,3-thia...)
Affinity DataIC50: 2.64E+3nMAssay Description:To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several c...More data for this Ligand-Target Pair
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PubMed
TargetTransmembrane protease serine 2(Human)
Fred Hutchinson Cancer Research Center

LigandPNGBDBM420292(4401-0077 | Antidepressant agent 1)
Affinity DataIC50: 2.68E+3nMAssay Description:To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several c...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In DepthDetails Article
PubMed