Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50045282
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055096(CHEMBL3317576)
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO cells assessed as inhibition of CCPA-stimulated cAMP level by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055099(CHEMBL3317579)
Affinity DataIC50: 2.90nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO cells assessed as inhibition of CCPA-stimulated cAMP level by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055098(CHEMBL3317578)
Affinity DataIC50: 4.30nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO cells assessed as inhibition of CCPA-stimulated cAMP level by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055095(CHEMBL3317575)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO cells assessed as inhibition of CCPA-stimulated cAMP level by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055094(CHEMBL3317574)
Affinity DataIC50: 43nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO cells assessed as inhibition of CCPA-stimulated cAMP level by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055087(CHEMBL3317565)
Affinity DataIC50: 123nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055098(CHEMBL3317578)
Affinity DataIC50: 247nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055099(CHEMBL3317579)
Affinity DataIC50: 314nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50427586(CHEMBL2322916)
Affinity DataIC50: 320nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055096(CHEMBL3317576)
Affinity DataIC50: 334nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055095(CHEMBL3317575)
Affinity DataIC50: 387nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50427584(CHEMBL2322918)
Affinity DataIC50: 420nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055094(CHEMBL3317574)
Affinity DataIC50: 423nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055094(CHEMBL3317574)
Affinity DataIC50: 432nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50427585(CHEMBL2322917)
Affinity DataIC50: 440nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055082(CHEMBL3317555)
Affinity DataIC50: 630nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP level by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055096(CHEMBL3317576)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055099(CHEMBL3317579)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055098(CHEMBL3317578)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055095(CHEMBL3317575)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055094(CHEMBL3317574)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055097(CHEMBL3317577)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055100(CHEMBL3317580)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055087(CHEMBL3317565)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055094(CHEMBL3317574)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055089(CHEMBL3317554)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50427586(CHEMBL2322916)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055084(CHEMBL3317559)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50427585(CHEMBL2322917)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055082(CHEMBL3317555)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055089(CHEMBL3317554)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055083(CHEMBL3317556)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055086(CHEMBL3317561)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055089(CHEMBL3317554)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]AB-MECA from human adenosine A3 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055098(CHEMBL3317578)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50427584(CHEMBL2322918)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055099(CHEMBL3317579)
Affinity DataKi:  146nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055096(CHEMBL3317576)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50427584(CHEMBL2322918)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055095(CHEMBL3317575)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055087(CHEMBL3317565)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055088(CHEMBL3317566)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055085(CHEMBL3317560)
Affinity DataKi:  213nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50427586(CHEMBL2322916)
Affinity DataKi:  246nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055090(CHEMBL3317568)
Affinity DataKi:  312nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50427585(CHEMBL2322917)
Affinity DataKi:  325nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055085(CHEMBL3317560)
Affinity DataKi:  375nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055092(CHEMBL3317572)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055082(CHEMBL3317555)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50055093(CHEMBL3317573)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
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