Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50006210
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497848(CHEMBL3319079)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497846(CHEMBL3319091)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497845(CHEMBL3319084)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497857(CHEMBL3319085)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497848(CHEMBL3319079)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497852(CHEMBL3319089)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497851(CHEMBL3319087)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497847(CHEMBL3319088)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497854(CHEMBL3319080)
Affinity DataKi:  314nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497855(CHEMBL3319081)
Affinity DataKi:  426nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497855(CHEMBL3319081)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497851(CHEMBL3319087)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497846(CHEMBL3319091)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497846(CHEMBL3319091)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497854(CHEMBL3319080)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497852(CHEMBL3319089)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497856(CHEMBL3319083)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497852(CHEMBL3319089)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497851(CHEMBL3319087)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497855(CHEMBL3319081)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497848(CHEMBL3319079)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497854(CHEMBL3319080)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497853(CHEMBL3319090)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497850(CHEMBL3319086)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497849(CHEMBL3319082)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497847(CHEMBL3319088)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50497847(CHEMBL3319088)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed