Compile Data Set for Download or QSAR
Report error Found 89 Enz. Inhib. hit(s) with all data for entry = 50045264
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053982(CHEMBL3319552)
Affinity DataEC50:  794nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053958(CHEMBL3319565)
Affinity DataEC50:  2.75E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053979(CHEMBL3319553)
Affinity DataEC50:  4.68E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053978(CHEMBL3319554)
Affinity DataEC50:  1.40E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053977(CHEMBL3319555)
Affinity DataEC50:  1.40E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053976(CHEMBL3319556)
Affinity DataEC50: >1.25E+4nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053975(CHEMBL3319557)
Affinity DataEC50:  1.15E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053974(CHEMBL3319558)
Affinity DataEC50:  416nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053971(CHEMBL3319559)
Affinity DataEC50:  351nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054054(CHEMBL3319547)
Affinity DataEC50:  2.95E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054053(CHEMBL3319548)
Affinity DataEC50:  933nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054052(CHEMBL3319549)
Affinity DataEC50:  205nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054051(CHEMBL3319550)
Affinity DataEC50:  1.29E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053983(CHEMBL3319551)
Affinity DataEC50: >1.25E+4nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053903(CHEMBL3319524)
Affinity DataEC50:  5.37E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054094(CHEMBL3319541)
Affinity DataEC50:  776nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054063(CHEMBL3319542)
Affinity DataEC50:  803nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054059(CHEMBL3319543)
Affinity DataEC50:  2.80E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054058(CHEMBL3317472)
Affinity DataEC50:  1.38E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054057(CHEMBL3319544)
Affinity DataEC50:  565nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054055(CHEMBL3319546)
Affinity DataEC50:  766nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054106(CHEMBL3319534)
Affinity DataEC50:  81nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054104(CHEMBL3319535)
Affinity DataEC50:  1.08E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054102(CHEMBL3319536)
Affinity DataEC50:  2.45E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054101(CHEMBL3319537)
Affinity DataEC50:  1.26E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054099(CHEMBL3319539)
Affinity DataEC50:  1.73E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054097(CHEMBL3319540)
Affinity DataEC50:  1.19E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054107(CHEMBL3319533)
Affinity DataEC50:  52nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053957(CHEMBL3319564)
Affinity DataEC50:  1.12E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053902(CHEMBL3319532)
Affinity DataEC50:  1.12E+4nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053950(CHEMBL3319527)
Affinity DataEC50:  3.35E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053951(CHEMBL3319528)
Affinity DataEC50:  510nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053952(CHEMBL3319529)
Affinity DataEC50:  254nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053953(CHEMBL3319530)
Affinity DataEC50:  2.14E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053954(CHEMBL3319531)
Affinity DataEC50:  2.00E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053959(CHEMBL3319522)
Affinity DataEC50: >1.25E+4nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053960(CHEMBL3319523)
Affinity DataEC50:  6.36E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053966(CHEMBL3319560)
Affinity DataEC50:  234nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053969(CHEMBL3319561)
Affinity DataEC50:  309nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Mouse)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053955(CHEMBL3319562)
Affinity DataEC50:  2.63E+3nMAssay Description:Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054107(CHEMBL3319533)
Affinity DataIC50: 1nMAssay Description:Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054052(CHEMBL3319549)
Affinity DataIC50: 5nMAssay Description:Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054106(CHEMBL3319534)
Affinity DataIC50: 5nMAssay Description:Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50053952(CHEMBL3319529)
Affinity DataIC50: 5nMAssay Description:Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054097(CHEMBL3319540)
Affinity DataIC50: 5nMAssay Description:Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054057(CHEMBL3319544)
Affinity DataIC50: 6nMAssay Description:Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054063(CHEMBL3319542)
Affinity DataIC50: 7nMAssay Description:Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054094(CHEMBL3319541)
Affinity DataIC50: 7nMAssay Description:Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054059(CHEMBL3319543)
Affinity DataIC50: 8nMAssay Description:Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50054058(CHEMBL3317472)
Affinity DataIC50: 11nMAssay Description:Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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