Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50045109
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434489(CHEMBL2385547)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045412(CHEMBL3314153)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045417(CHEMBL3314148)
Affinity DataIC50: 13nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045423(CHEMBL3314142)
Affinity DataIC50: 14nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045418(CHEMBL3314147)
Affinity DataIC50: 16nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045416(CHEMBL3314149)
Affinity DataIC50: 17nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045415(CHEMBL3314150)
Affinity DataIC50: 22nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045422(CHEMBL3314143)
Affinity DataIC50: 23nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045373(CHEMBL3315291)
Affinity DataIC50: 25nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045371(CHEMBL3315292)
Affinity DataIC50: 26nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 26nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045409(CHEMBL3314156)
Affinity DataIC50: 26nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045374(CHEMBL3315290)
Affinity DataIC50: 26nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045414(CHEMBL3314151)
Affinity DataIC50: 31nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045411(CHEMBL3314154)
Affinity DataIC50: 36nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045410(CHEMBL3314155)
Affinity DataIC50: 37nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045413(CHEMBL3314152)
Affinity DataIC50: 44nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045399(CHEMBL3315287)
Affinity DataIC50: 55nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045404(CHEMBL3315286)
Affinity DataIC50: 65nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045385(CHEMBL3315289)
Affinity DataIC50: 67nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045394(CHEMBL3315288)
Affinity DataIC50: 75nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045425(CHEMBL3314141)
Affinity DataIC50: 85nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045419(CHEMBL3314146)
Affinity DataIC50: 95nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045421(CHEMBL3314144)
Affinity DataIC50: 157nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045407(CHEMBL3314157)
Affinity DataIC50: 160nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045420(CHEMBL3314145)
Affinity DataIC50: 450nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as reduction in LPS-induced HSP27 Ser78 phosphorylation after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045405(CHEMBL3315285)
Affinity DataIC50: 3.39E+3nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045406(CHEMBL3314158)
Affinity DataIC50: 3.73E+3nMAssay Description:Inhibition of MK2 (unknown origin) incubated for 30 mins by MK2 IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of AKT1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ROCK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInsulin-like growth factor 1 receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of IGF1R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalcium/calmodulin-dependent protein kinase type IV(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CAMK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of GSK3B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEphrin type-B receptor 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of EPHB4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of RSK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of IKKB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CHK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of IRAK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha type(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PKCA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of LCK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of NEK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CSNK1D (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 3(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MST2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PLK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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