Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50043681
TargetBile salt export pump(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444583(CHEMBL3099716 | US9340549, 74)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of BSEP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444583(CHEMBL3099716 | US9340549, 74)
Affinity DataIC50: 4.85E+4nMAssay Description:Binding affinity to NK1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444583(CHEMBL3099716 | US9340549, 74)
Affinity DataIC50: 4.85E+4nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444583(CHEMBL3099716 | US9340549, 74)
Affinity DataIC50: 4.85E+4nMAssay Description:Binding affinity to dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444583(CHEMBL3099716 | US9340549, 74)
Affinity DataIC50: 4.85E+4nMAssay Description:Binding affinity to CCR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444584(CHEMBL3099718 | US9340549, 95)
Affinity DataIC50: 8.50E+4nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444583(CHEMBL3099716 | US9340549, 74)
Affinity DataIC50: 8.50E+4nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444585(CHEMBL3099720 | US9340549, 65)
Affinity DataIC50: 8.50E+4nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 2(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444584(CHEMBL3099718 | US9340549, 95)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 2(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444583(CHEMBL3099716 | US9340549, 74)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 2(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50444585(CHEMBL3099720 | US9340549, 65)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed