Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50039810
LigandPNGBDBM50384542(CHEMBL2036616)
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50362106(CHEMBL1938681)
Affinity DataEC50:  350nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384542(CHEMBL2036616)
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384544(CHEMBL2036610)
Affinity DataEC50:  760nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384572(CHEMBL2036606)
Affinity DataEC50:  730nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384570(CHEMBL2036604)
Affinity DataEC50:  820nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384567(CHEMBL2036601)
Affinity DataEC50:  2.40E+3nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384562(CHEMBL2036459)
Affinity DataEC50:  3.70E+3nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384561(CHEMBL2036458)
Affinity DataEC50:  2.70E+3nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384559(CHEMBL2036456)
Affinity DataEC50:  3.00E+3nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384555(CHEMBL2036452)
Affinity DataEC50:  6.70E+3nMAssay Description:Inhibition of MK2 in human THP1 cells assessed as inhibition of LPS-induced HSP27 Ser78 phosphorylation incubated for 60 mins prior to LPS-induction ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384542(CHEMBL2036616)
Affinity DataIC50: 6nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50384542(CHEMBL2036616)
Affinity DataIC50: 8nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384542(CHEMBL2036616)
Affinity DataIC50: 8nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384561(CHEMBL2036458)
Affinity DataIC50: 30nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384559(CHEMBL2036456)
Affinity DataIC50: 30nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384572(CHEMBL2036606)
Affinity DataIC50: 40nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384555(CHEMBL2036452)
Affinity DataIC50: 50nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384560(CHEMBL2036457)
Affinity DataIC50: 50nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384544(CHEMBL2036610)
Affinity DataIC50: 50nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384575(CHEMBL2036460)
Affinity DataIC50: 60nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384562(CHEMBL2036459)
Affinity DataIC50: 60nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384563(CHEMBL2036461)
Affinity DataIC50: 70nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384567(CHEMBL2036601)
Affinity DataIC50: 70nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384570(CHEMBL2036604)
Affinity DataIC50: 100nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384565(CHEMBL2036599)
Affinity DataIC50: 100nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384557(CHEMBL2036454)
Affinity DataIC50: 110nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50362106(CHEMBL1938681)
Affinity DataIC50: 110nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384564(CHEMBL2036598)
Affinity DataIC50: 160nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384573(CHEMBL2036607)
Affinity DataIC50: 180nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384551(CHEMBL2036618)
Affinity DataIC50: 190nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384566(CHEMBL2036600)
Affinity DataIC50: 190nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384546(CHEMBL2036612)
Affinity DataIC50: 220nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384548(CHEMBL2036614)
Affinity DataIC50: 310nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384569(CHEMBL2036603)
Affinity DataIC50: 330nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384571(CHEMBL2036605)
Affinity DataIC50: 380nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384574(CHEMBL2036608)
Affinity DataIC50: 480nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384547(CHEMBL2036613)
Affinity DataIC50: 790nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384545(CHEMBL2036611)
Affinity DataIC50: 970nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384568(CHEMBL2036602)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384543(CHEMBL2036609)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384558(CHEMBL2036455)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384552(CHEMBL2036449)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384556(CHEMBL2036453)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384550(CHEMBL2036617)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384554(CHEMBL2036451)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384541(CHEMBL2036620)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384549(CHEMBL2036615)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384540(CHEMBL2036619)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50384553(CHEMBL2036450)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MK2 using 5TAMRA-KKLNRTLSVA-COOH as substrate incubated for 30 mins prior to substrate addition measured after 30 mins by immobilized m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed