Compile Data Set for Download or QSAR
Report error Found 333 Enz. Inhib. hit(s) with all data for entry = 50045090
TargetVasopressin V2 receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044676(CHEMBL439044)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at human vasopressin V2 expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human vasopressin V2 expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  7.30nMAssay Description:Agonist activity at human vasopressin V2 expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044678(CHEMBL3354602)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044679(CHEMBL3354601)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044680(CHEMBL3354600)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044681(CHEMBL3354599)
Affinity DataEC50:  0.780nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044682(CHEMBL3354598)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044683(CHEMBL3354597)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044684(CHEMBL3354596)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044685(CHEMBL3354595)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044686(CHEMBL3354594)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044687(CHEMBL3354593)
Affinity DataEC50:  0.560nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044727(CHEMBL3354592)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044728(CHEMBL3354591)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044729(CHEMBL3354590)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044730(CHEMBL3354589)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044731(CHEMBL3354588)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044732(CHEMBL3354587)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044733(CHEMBL3354586)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044734(CHEMBL3354585)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044735(CHEMBL3354584)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044736(CHEMBL3354583)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044737(CHEMBL3354582)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044738(CHEMBL3354581)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044740(CHEMBL3352839)
Affinity DataEC50:  0.860nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044741(CHEMBL3354580)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044742(CHEMBL3354579)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044743(CHEMBL3354578)
Affinity DataEC50:  0.850nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044744(CHEMBL3354577)
Affinity DataEC50:  0.960nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044745(CHEMBL3354576)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044746(CHEMBL3354575)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044747(CHEMBL3354574)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044748(CHEMBL3354573)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044749(CHEMBL3354572)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044750(CHEMBL3354571)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044751(CHEMBL3354570)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044752(CHEMBL3353956)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044754(CHEMBL3353955)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044755(CHEMBL3353954)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044756(CHEMBL3353953)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044757(CHEMBL3353952)
Affinity DataEC50:  0.460nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044758(CHEMBL3353951)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044759(CHEMBL3353950)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044760(CHEMBL3353949)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044761(CHEMBL3353948)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044762(CHEMBL3353947)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044763(CHEMBL3353946)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044764(CHEMBL3353945)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50044765(CHEMBL3353944)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human oxytocin receptor expressed in CHO-K1 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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