Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50044592
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of DYRK1A (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of DYRK1A (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:Inhibition of CDK5 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of rat DYRK1A assessed as inhibition of phosphate incorporation using GRSRSRSRSRSR and [gamma-33P]ATP as substrate after 30 mins by scinti...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of CLK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mouse)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of mouse recombinant GST-fused CLK1 expressed in Escherichia coli cells assessed as inhibition of phosphate incorporation using GRSRSRSRSR...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of CDK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Inhibition of CDK9/cyclin T (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of DYRK3 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of DYRK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of CLK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK3(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of CLK3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of CDK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of CLK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of CDK5 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin) assessed as inhibition of phosphate incorporation using histone 1 and [gamma-33P]ATP as substrate after 30 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK5 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK5 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK5 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
