Compile Data Set for Download or QSAR
Report error Found 151 Enz. Inhib. hit(s) with all data for entry = 50044401
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50016165(CHEMBL3261516)
Affinity DataIC50: 6nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016166(CHEMBL3261517)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 10nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 2 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 10nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 1 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 13nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 6 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50016148(CHEMBL3261500)
Affinity DataIC50: 14nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 14nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.667 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 17nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.012 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50016160(CHEMBL3261511)
Affinity DataIC50: 18nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016161(CHEMBL3261512)
Affinity DataIC50: 18nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 18nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 9 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 20nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.333 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50016167(CHEMBL3261518)
Affinity DataIC50: 21nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 23nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 18 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 29nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.111 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50016162(CHEMBL3261513)
Affinity DataIC50: 33nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 35nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.222 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 40nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.025 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50016153(CHEMBL3261505)
Affinity DataIC50: 42nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 44nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 27 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016164(CHEMBL3261515)
Affinity DataIC50: 62nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 63nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.037 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 64nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.074 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform delta(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 84nMAssay Description:Inhibition of CK1delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 86nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 54 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016147(CHEMBL3261499)
Affinity DataIC50: 96nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016137(CHEMBL3261489)
Affinity DataIC50: 101nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016146(CHEMBL3261498)
Affinity DataIC50: 104nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform delta(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50016166(CHEMBL3261517)
Affinity DataIC50: 104nMAssay Description:Inhibition of CK1delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016136(CHEMBL3261488)
Affinity DataIC50: 115nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016135(CHEMBL3261245)
Affinity DataIC50: 172nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016116(CHEMBL3261228)
Affinity DataIC50: 300nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.023 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016116(CHEMBL3261228)
Affinity DataIC50: 316nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.75 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016116(CHEMBL3261228)
Affinity DataIC50: 318nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 1.5 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016116(CHEMBL3261228)
Affinity DataIC50: 323nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016116(CHEMBL3261228)
Affinity DataIC50: 405nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.047 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016116(CHEMBL3261228)
Affinity DataIC50: 419nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 3 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016129(CHEMBL3261240)
Affinity DataIC50: 451nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016144(CHEMBL3261496)
Affinity DataIC50: 452nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016141(CHEMBL3261493)
Affinity DataIC50: 472nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 501nMAssay Description:Inhibition of Cdc7/Dbf4 in human HCT116 cells assessed as reduction of MCM2 phosphorylation after 14 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016116(CHEMBL3261228)
Affinity DataIC50: 528nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.094 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016127(CHEMBL3261238)
Affinity DataIC50: 529nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform alpha(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50016166(CHEMBL3261517)
Affinity DataIC50: 545nMAssay Description:Inhibition of CK1alpha (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016116(CHEMBL3261228)
Affinity DataIC50: 546nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.375 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016116(CHEMBL3261228)
Affinity DataIC50: 547nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.188 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016122(CHEMBL3261234)
Affinity DataIC50: 669nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform alpha(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50: 694nMAssay Description:Inhibition of CK1alpha (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50016148(CHEMBL3261500)
Affinity DataIC50: 700nMAssay Description:Inhibition of CDK2/Cyclin-E (unknown origin) using maltose binding protein as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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