Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50044295
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011716(CHEMBL3262896)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at EBI2 receptor in human U937 cells assessed as inhibition of 7-alpha,25-OHC-induced cell migration after 3 hrs by flow cytometr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011701(CHEMBL3262895)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011717(CHEMBL3262876)
Affinity DataIC50: 5.30nMAssay Description:Antagonist activity at EBI2 receptor in human U937 cells assessed as inhibition of 7-alpha,25-OHC-induced cell migration after 3 hrs by flow cytometr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011701(CHEMBL3262895)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011716(CHEMBL3262896)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of 0.1 nM oxysterol-induced [35S]GTPgammaS bindi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011716(CHEMBL3262896)
Affinity DataIC50: 8.5nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of 0.33 nM oxysterol-induced [35S]GTPgammaS bind...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011716(CHEMBL3262896)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at EBI2 receptor in human U937 cells assessed as inhibition of oxysterol-induced calcium release measured for 3 mins by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011716(CHEMBL3262896)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011689(CHEMBL3262892)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011716(CHEMBL3262896)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011692(CHEMBL3262894)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011725(CHEMBL3262883)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011578(CHEMBL3262890)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011578(CHEMBL3262890)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011592(CHEMBL3262891)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011722(CHEMBL3262880)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011731(CHEMBL3262889)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011731(CHEMBL3262889)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011721(CHEMBL3262879)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011689(CHEMBL3262892)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011692(CHEMBL3262894)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011724(CHEMBL3262882)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011719(CHEMBL3262877)
Affinity DataIC50: 28nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011721(CHEMBL3262879)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011592(CHEMBL3262891)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011723(CHEMBL3262881)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011726(CHEMBL3262884)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011730(CHEMBL3262888)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011729(CHEMBL3262887)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011724(CHEMBL3262882)
Affinity DataIC50: 44nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011690(CHEMBL3262893)
Affinity DataIC50: 44nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011725(CHEMBL3262883)
Affinity DataIC50: 46nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011690(CHEMBL3262893)
Affinity DataIC50: 52nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011730(CHEMBL3262888)
Affinity DataIC50: 55nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011729(CHEMBL3262887)
Affinity DataIC50: 65nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011728(CHEMBL3262886)
Affinity DataIC50: 68nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011727(CHEMBL3262885)
Affinity DataIC50: 81nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011717(CHEMBL3262876)
Affinity DataIC50: 83nMAssay Description:Displacement of [3H]-7-alpha,25-OHC from recombinant human EBI2 receptor expressed in CHO cells after 10 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011726(CHEMBL3262884)
Affinity DataIC50: 84nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011722(CHEMBL3262880)
Affinity DataIC50: 91nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011717(CHEMBL3262876)
Affinity DataIC50: 91nMAssay Description:Antagonist activity at EBI2 receptor in human U937 cells assessed as inhibition of oxysterol-induced calcium release measured for 3 mins by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011728(CHEMBL3262886)
Affinity DataIC50: 92nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011727(CHEMBL3262885)
Affinity DataIC50: 98nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011719(CHEMBL3262877)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011717(CHEMBL3262876)
Affinity DataIC50: 196nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011723(CHEMBL3262881)
Affinity DataIC50: 209nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011718(CHEMBL1305842)
Affinity DataIC50: 309nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011717(CHEMBL3262876)
Affinity DataIC50: 423nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011718(CHEMBL1305842)
Affinity DataIC50: 977nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 183(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011720(CHEMBL3262878)
Affinity DataIC50: 2.95E+3nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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