Compile Data Set for Download or QSAR
Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 50043617
LigandPNGBDBM50443648(CHEMBL3093076)
Affinity DataIC50: 0.690nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443649(CHEMBL3093075)
Affinity DataIC50: 0.850nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443650(CHEMBL3093074)
Affinity DataIC50: 1nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443644(CHEMBL3093080)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443646(CHEMBL3093078)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443647(CHEMBL3093077)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443651(CHEMBL3093073)
Affinity DataIC50: 2nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443645(CHEMBL3093079)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443652(CHEMBL3093072)
Affinity DataIC50: 4nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443653(CHEMBL3093071)
Affinity DataIC50: 7nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443642(CHEMBL3093056)
Affinity DataIC50: 10nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443660(CHEMBL3093064)
Affinity DataIC50: 10nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443665(CHEMBL3093059)
Affinity DataIC50: 11nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443643(CHEMBL3093055)
Affinity DataIC50: 17nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443649(CHEMBL3093075)
Affinity DataIC50: 20nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443666(CHEMBL3093058)
Affinity DataIC50: 20nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443662(CHEMBL3093062)
Affinity DataIC50: 24nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443659(CHEMBL3093065)
Affinity DataIC50: 25nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50443649(CHEMBL3093075)
Affinity DataIC50: 31nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using 4eBP1 ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443644(CHEMBL3093080)
Affinity DataIC50: 32nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443654(CHEMBL3093070)
Affinity DataIC50: 32nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443655(CHEMBL3093069)
Affinity DataIC50: 35nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443661(CHEMBL3093063)
Affinity DataIC50: 35nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443648(CHEMBL3093076)
Affinity DataIC50: 51nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443647(CHEMBL3093077)
Affinity DataIC50: 60nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443660(CHEMBL3093064)
Affinity DataIC50: 61nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443650(CHEMBL3093074)
Affinity DataIC50: 71nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443655(CHEMBL3093069)
Affinity DataIC50: 98nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443659(CHEMBL3093065)
Affinity DataIC50: 98nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443656(CHEMBL3093068)
Affinity DataIC50: 110nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443653(CHEMBL3093071)
Affinity DataIC50: 120nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50443648(CHEMBL3093076)
Affinity DataIC50: 120nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using 4eBP1 ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443646(CHEMBL3093078)
Affinity DataIC50: 130nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443651(CHEMBL3093073)
Affinity DataIC50: 140nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443662(CHEMBL3093062)
Affinity DataIC50: 150nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443652(CHEMBL3093072)
Affinity DataIC50: 150nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443666(CHEMBL3093058)
Affinity DataIC50: 170nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443658(CHEMBL3093066)
Affinity DataIC50: 170nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443657(CHEMBL3093067)
Affinity DataIC50: 190nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated MCM2 phosphorylation at Ser53 by protein A amplified luminescent proximity homogeneous assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443665(CHEMBL3093059)
Affinity DataIC50: 230nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443649(CHEMBL3093075)
Affinity DataIC50: 240nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443645(CHEMBL3093079)
Affinity DataIC50: 250nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443654(CHEMBL3093070)
Affinity DataIC50: 310nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443656(CHEMBL3093068)
Affinity DataIC50: 350nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443643(CHEMBL3093055)
Affinity DataIC50: 350nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443654(CHEMBL3093070)
Affinity DataIC50: 370nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50443644(CHEMBL3093080)
Affinity DataIC50: 460nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using 4eBP1 ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443648(CHEMBL3093076)
Affinity DataIC50: 490nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443660(CHEMBL3093064)
Affinity DataIC50: 580nMAssay Description:Inhibition of Cdc7-mediated MCM2 phosphorylation at Ser53 in human HCT116 cells after 14 hrs by immunostaining assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50443661(CHEMBL3093063)
Affinity DataIC50: 580nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using ULight peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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