Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50001513
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataIC50: 1.30nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataIC50: 21nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016013(6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quino...)
Affinity DataIC50: 58nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016013(6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quino...)
Affinity DataIC50: 107nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016017(Quinerolane | (5aR,9aR)-6-propyl-5,5a,6,7,8,9,9a,1...)
Affinity DataIC50: 151nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016011(CHEMBL155884 | (R)-10-bromo-6-methyl-5,6,6a,7-tetr...)
Affinity DataIC50: 171nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016010(CHEMBL155833 | 8-Bromo-6-methyl-5,6,6a,7-tetrahydr...)
Affinity DataIC50: 181nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataIC50: 432nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016010(CHEMBL155833 | 8-Bromo-6-methyl-5,6,6a,7-tetrahydr...)
Affinity DataIC50: 449nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016006(CHEMBL153960 | 8-Chloro-6-methyl-5,6,6a,7-tetrahyd...)
Affinity DataIC50: 500nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016006(CHEMBL153960 | 8-Chloro-6-methyl-5,6,6a,7-tetrahyd...)
Affinity DataIC50: 561nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016016(CHEMBL345907 | 10-Chloro-6-methyl-5,6,6a,7-tetrahy...)
Affinity DataIC50: 637nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016011(CHEMBL155884 | (R)-10-bromo-6-methyl-5,6,6a,7-tetr...)
Affinity DataIC50: 664nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM29643(CHEMBL416288 | Apomorphine,(+) | (S)-6-methyl-5,6,...)
Affinity DataIC50: 680nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016018((S)-11-methoxy-7-methyl-6,7,7a,8-tetrahydro-5H-ben...)
Affinity DataIC50: 739nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016016(CHEMBL345907 | 10-Chloro-6-methyl-5,6,6a,7-tetrahy...)
Affinity DataIC50: 803nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016020(CHEMBL154989 | 9-Bromo-6-methyl-5,6,6a,7-tetrahydr...)
Affinity DataIC50: 818nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016014(CHEMBL155246 | 11-Methoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50: 829nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016012(CHEMBL155883 | 8,10-Dibromo-6-methyl-5,6,6a,7-tetr...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016015(CHEMBL157735 | 9-Bromo-6-methyl-5,6,6a,7-tetrahydr...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016015(CHEMBL157735 | 9-Bromo-6-methyl-5,6,6a,7-tetrahydr...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016012(CHEMBL155883 | 8,10-Dibromo-6-methyl-5,6,6a,7-tetr...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016019(CHEMBL154709 | 10-Methoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50: 2.08E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016007(CHEMBL117841 | 11-Methoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50: 2.16E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016005(CHEMBL157879 | 6-Methyl-5,6,6a,7-tetrahydro-4H-dib...)
Affinity DataIC50: 2.24E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016020(CHEMBL154989 | 9-Bromo-6-methyl-5,6,6a,7-tetrahydr...)
Affinity DataIC50: 2.58E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016009(CHEMBL345822 | 10-Bromo-6-methyl-5,6,6a,7-tetrahyd...)
Affinity DataIC50: 2.93E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016007(CHEMBL117841 | 11-Methoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50: 3.28E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016009(CHEMBL345822 | 10-Bromo-6-methyl-5,6,6a,7-tetrahyd...)
Affinity DataIC50: 3.34E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM29643(CHEMBL416288 | Apomorphine,(+) | (S)-6-methyl-5,6,...)
Affinity DataIC50: 3.62E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016005(CHEMBL157879 | 6-Methyl-5,6,6a,7-tetrahydro-4H-dib...)
Affinity DataIC50: 5.06E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016008(CHEMBL346017 | 8-Bromo-6-methyl-5,6,6a,7-tetrahydr...)
Affinity DataIC50: 8.61E+3nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016017(Quinerolane | (5aR,9aR)-6-propyl-5,5a,6,7,8,9,9a,1...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016008(CHEMBL346017 | 8-Bromo-6-methyl-5,6,6a,7-tetrahydr...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016014(CHEMBL155246 | 11-Methoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50: 1.21E+4nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016019(CHEMBL154709 | 10-Methoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataIC50: 1.33E+4nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]SCH-23390 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50016018((S)-11-methoxy-7-methyl-6,7,7a,8-tetrahydro-5H-ben...)
Affinity DataIC50: 1.40E+4nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed