Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50005595
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50392637(CHEMBL215421)
Affinity DataKi:  0.407nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493054(CHEMBL2419769)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50392637(CHEMBL215421)
Affinity DataKi:  0.513nMAssay Description:Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50411188(CHEMBL217469)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50026917(CHEMBL13647 | BMY 7378 | 8-{2-[4-(2-Methoxy-phenyl...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to human 5-HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493054(CHEMBL2419769)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493056(CHEMBL2419771)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493056(CHEMBL2419771)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50392637(CHEMBL215421)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493054(CHEMBL2419769)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493055(CHEMBL3216590)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50392637(CHEMBL215421)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50411188(CHEMBL217469)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493058(CHEMBL2419770)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493058(CHEMBL2419770)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50411188(CHEMBL217469)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493055(CHEMBL3216590)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50411188(CHEMBL217469)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493053(CHEMBL2419772)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493058(CHEMBL2419770)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493053(CHEMBL2419772)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493056(CHEMBL2419771)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493054(CHEMBL2419769)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493059(CHEMBL3217244)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493055(CHEMBL3216590)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493056(CHEMBL2419771)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493059(CHEMBL3217244)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493055(CHEMBL3216590)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493058(CHEMBL2419770)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493053(CHEMBL2419772)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493053(CHEMBL2419772)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493052(CHEMBL2419765)
Affinity DataKi:  178nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493059(CHEMBL3217244)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50099326(SNAP-8719 | 8-{(S)-1-Methyl-2-[4-(2,4,5-trifluoro-...)
Affinity DataKi:  302nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493052(CHEMBL2419765)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493059(CHEMBL3217244)
Affinity DataKi:  372nMAssay Description:Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493057(CHEMBL2419766)
Affinity DataKi:  437nMAssay Description:Displacement of [3H]prazosin from human alpha-1A adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493052(CHEMBL2419765)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493052(CHEMBL2419765)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493057(CHEMBL2419766)
Affinity DataKi:  1.35E+3nMAssay Description:Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493057(CHEMBL2419766)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50493057(CHEMBL2419766)
Affinity DataKi:  1.91E+3nMAssay Description:Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed