Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50005617
Affinity DataEC50: 17nMAssay Description:Antagonist activity at CB2 receptor in HEK293 cells assessed as increase in CP-55,940 EC50 measuring inhibition of forskolin-stimulated cAMP accumula...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Antagonist activity at CB2 receptor in HEK293 cells assessed as increase in CP-55,940 EC50 measuring inhibition of forskolin-stimulated cAMP accumula...More data for this Ligand-Target Pair
Affinity DataEC50: 5.30nMAssay Description:Antagonist activity at CB2 receptor in HEK293 cells assessed as increase in CP-55,940 EC50 measuring inhibition of forskolin-stimulated cAMP accumula...More data for this Ligand-Target Pair
Affinity DataEC50: 4.20nMAssay Description:Agonist activity at CB2 receptor in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulationMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataEC50: 43nMAssay Description:Antagonist activity at CB2 receptor in HEK293 cells assessed as increase in CP-55,940 EC50 measuring inhibition of forskolin-stimulated cAMP accumula...More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Antagonist activity at CB2 receptor in HEK293 cells assessed as increase in CP-55,940 EC50 measuring inhibition of forskolin-stimulated cAMP accumula...More data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Antagonist activity at CB2 receptor in HEK293 cells assessed as increase in CP-55,940 EC50 measuring inhibition of forskolin-stimulated cAMP accumula...More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 527nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.22E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
