Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50043276
TargetD(2) dopamine receptor(Human)
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM50438565(CHEMBL2413153)
Affinity DataKi:  37nMAssay Description:Binding affinity to dopamine 2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM86757(NSC_11603174 | CAS_0 | [11C]MMP)
Affinity DataKi:  59nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM50438565(CHEMBL2413153)
Affinity DataKi:  512nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM86757(NSC_11603174 | CAS_0 | [11C]MMP)
Affinity DataKi:  1.03E+3nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistamine H2 receptor(Human)
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM50438565(CHEMBL2413153)
Affinity DataKi:  1.77E+3nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistamine H2 receptor(Human)
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM86757(NSC_11603174 | CAS_0 | [11C]MMP)
Affinity DataKi:  2.13E+3nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM50438565(CHEMBL2413153)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM86757(NSC_11603174 | CAS_0 | [11C]MMP)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to dopamine 2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed