Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50043274
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438555(CHEMBL2413142)
Affinity DataIC50: 32nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438554(CHEMBL2413143)
Affinity DataIC50: 35nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438549(CHEMBL2413146)
Affinity DataIC50: 50nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438562(CHEMBL2413135)
Affinity DataIC50: 72nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438560(CHEMBL2413137)
Affinity DataIC50: 100nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438553(CHEMBL2413144)
Affinity DataIC50: 140nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438561(CHEMBL2413136)
Affinity DataIC50: 300nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438556(CHEMBL2413141)
Affinity DataIC50: 370nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438552(CHEMBL2413145)
Affinity DataIC50: 540nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438550(CHEMBL2413133)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of ATPase activity of CENP-E motor domain (unknown origin) by high throughput screening assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438550(CHEMBL2413133)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438563(CHEMBL2413134)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438557(CHEMBL2413140)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438551(CHEMBL2413132)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of ATPase activity of CENP-E motor domain (unknown origin) by high throughput screening assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438558(CHEMBL2413139)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCentromere-associated protein E(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50438559(CHEMBL2413138)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of human ATPase activity of CENP-E motor domain assessed as ADP production after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed