Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50005500
TargetMu-type opioid/Nociceptin receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50492400(CHEMBL2403214)
Affinity DataEC50:  316nMAssay Description:Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50492401(CHEMBL2403215)
Affinity DataEC50:  1.62E+3nMAssay Description:Activity at Wistar rat mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of nal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetNociceptin receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50492402(CHEMBL2403216)
Affinity DataEC50:  1.66E+3nMAssay Description:Activity at Wistar rat NOP receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of naloxoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetNociceptin receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM85191(CAS_200959-47-3 | Ac-RYYRWK-NH2)
Affinity DataEC50:  6.20nMAssay Description:Activity at Wistar rat NOP receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of naloxoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50492401(CHEMBL2403215)
Affinity DataEC50:  1.23E+3nMAssay Description:Activity at Wistar rat mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetMu-type opioid/Nociceptin receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50492403(CHEMBL2403213)
Affinity DataEC50:  550nMAssay Description:Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetMu-type opioid/Nociceptin receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50492400(CHEMBL2403214)
Affinity DataEC50:  617nMAssay Description:Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetNociceptin receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50106479(FGGFTGARKSARK | H-FGGFTGARKSARK-NH2 | NC(1-13)NH2 ...)
Affinity DataEC50:  51nMAssay Description:Activity at Wistar rat NOP receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetNociceptin receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50492402(CHEMBL2403216)
Affinity DataEC50:  1.41E+3nMAssay Description:Activity at Wistar rat NOP receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50492404(CHEMBL2403217)
Affinity DataEC50:  1.02E+3nMAssay Description:Activity at Wistar rat mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50492404(CHEMBL2403217)
Affinity DataEC50:  1.15E+3nMAssay Description:Activity at Wistar rat mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contraction in presence of nal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetMu-type opioid/Nociceptin receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50492403(CHEMBL2403213)
Affinity DataEC50:  1.66E+3nMAssay Description:Activity at Wistar rat NOP/mu opioid receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetNociceptin receptor(Rat)
Bulgarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM85191(CAS_200959-47-3 | Ac-RYYRWK-NH2)
Affinity DataEC50:  16nMAssay Description:Activity at Wistar rat NOP receptor assessed as inhibition of low-frequency electrically-stimulated vas deferens contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed