Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 5995
TargetLysine-specific demethylase 4E(Human)
University of Oxford

LigandPNGBDBM50193145(Isoquinoline 3 | CHEMBL426560 | N-[(1-CHLORO-4-HYD...)
Affinity DataIC50: 2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 3A(Human)
University of Oxford

LigandPNGBDBM50193145(Isoquinoline 3 | CHEMBL426560 | N-[(1-CHLORO-4-HYD...)
Affinity DataIC50: 2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A [1-973](Human)
University of Oxford

LigandPNGBDBM50193145(Isoquinoline 3 | CHEMBL426560 | N-[(1-CHLORO-4-HYD...)
Affinity DataIC50: 2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Oxford

LigandPNGBDBM50193145(Isoquinoline 3 | CHEMBL426560 | N-[(1-CHLORO-4-HYD...)
Affinity DataIC50: 2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 2A(Human)
University of Oxford

LigandPNGBDBM50193145(Isoquinoline 3 | CHEMBL426560 | N-[(1-CHLORO-4-HYD...)
Affinity DataIC50: 2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4C [1-973](Human)
University of Oxford

LigandPNGBDBM50193145(Isoquinoline 3 | CHEMBL426560 | N-[(1-CHLORO-4-HYD...)
Affinity DataIC50: 2.00E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A [1-973](Human)
University of Oxford

LigandPNGBDBM103845(4HQ derivative 8)
Affinity DataIC50: 4.30E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 2A(Human)
University of Oxford

LigandPNGBDBM103843(4HQ derivative 6)
Affinity DataIC50: 5.20E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4C [1-973](Human)
University of Oxford

LigandPNGBDBM103845(4HQ derivative 8)
Affinity DataIC50: 8.60E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4C [1-973](Human)
University of Oxford

LigandPNGBDBM103846(4HQ derivative 9)
Affinity DataIC50: 9.30E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

LigandPNGBDBM103845(4HQ derivative 8)
Affinity DataIC50: 9.90E+4nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 3A(Human)
University of Oxford

LigandPNGBDBM103846(4HQ derivative 9)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 5C(Human)
University of Oxford

LigandPNGBDBM103846(4HQ derivative 9)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 2A(Human)
University of Oxford

LigandPNGBDBM103846(4HQ derivative 9)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 3A(Human)
University of Oxford

LigandPNGBDBM103842(4HQ derivative 4)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 3A(Human)
University of Oxford

LigandPNGBDBM103843(4HQ derivative 6)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 3A(Human)
University of Oxford

LigandPNGBDBM103844(4HQ derivative 7)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 2A(Human)
University of Oxford

LigandPNGBDBM103845(4HQ derivative 8)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 3A(Human)
University of Oxford

LigandPNGBDBM103845(4HQ derivative 8)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Oxford

LigandPNGBDBM103845(4HQ derivative 8)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 2A(Human)
University of Oxford

LigandPNGBDBM103842(4HQ derivative 4)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 2A(Human)
University of Oxford

LigandPNGBDBM103844(4HQ derivative 7)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4C [1-973](Human)
University of Oxford

LigandPNGBDBM103842(4HQ derivative 4)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A [1-973](Human)
University of Oxford

LigandPNGBDBM103842(4HQ derivative 4)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A [1-973](Human)
University of Oxford

LigandPNGBDBM103843(4HQ derivative 6)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A [1-973](Human)
University of Oxford

LigandPNGBDBM103844(4HQ derivative 7)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Oxford

LigandPNGBDBM103846(4HQ derivative 9)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4C [1-973](Human)
University of Oxford

LigandPNGBDBM103843(4HQ derivative 6)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4C [1-973](Human)
University of Oxford

LigandPNGBDBM103844(4HQ derivative 7)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

LigandPNGBDBM103842(4HQ derivative 4)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

LigandPNGBDBM103843(4HQ derivative 6)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

LigandPNGBDBM103844(4HQ derivative 7)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Oxford

LigandPNGBDBM103842(4HQ derivative 4)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Oxford

LigandPNGBDBM103843(4HQ derivative 6)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Oxford

LigandPNGBDBM103844(4HQ derivative 7)
Affinity DataIC50: 1.00E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 5C(Human)
University of Oxford

LigandPNGBDBM103845(4HQ derivative 8)
Affinity DataIC50: 1.23E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 5C(Human)
University of Oxford

LigandPNGBDBM103843(4HQ derivative 6)
Affinity DataIC50: 1.59E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 5C(Human)
University of Oxford

LigandPNGBDBM103842(4HQ derivative 4)
Affinity DataIC50: 4.43E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 5C(Human)
University of Oxford

LigandPNGBDBM103844(4HQ derivative 7)
Affinity DataIC50: 4.65E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed
TargetLysine-specific demethylase 5C(Human)
University of Oxford

LigandPNGBDBM50193145(Isoquinoline 3 | CHEMBL426560 | N-[(1-CHLORO-4-HYD...)
Affinity DataIC50: 5.50E+5nMpH: 7.5Assay Description:Inhibition assays were carried out in 384-well white ProxiPlates(PerkinElmer) in 10 μL of reaction volume. Standard reaction mixturesconsisted o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2014
Entry Details Article
PubMed