Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50005449
TargetAmyloid-beta precursor protein(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50485236(CHEBI:79033 | BAY-949172 | Florbetaben (18f) | Flo...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]IMPY from amyloid beta in brain homogenate of Alzheimer's disease patient after 2 hrs by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50484946(CHEBI:66880 | (18F)AV-45 | 18F-AV-45 | AV-45 F-18 ...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]IMPY from amyloid beta in brain homogenate of Alzheimer's disease patient after 2 hrs by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50122787(4-(6-iodoimidazo[1,2-a]pyridin-2-yl)-N,N-dimethyla...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]IMPY from amyloid beta (1 to 42) (unknown origin) after 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50122787(4-(6-iodoimidazo[1,2-a]pyridin-2-yl)-N,N-dimethyla...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]IMPY from amyloid beta (1 to 40) (unknown origin) after 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50492183(CHEMBL2397721)
Affinity DataKi:  28nMAssay Description:Displacement of [125I]IMPY from amyloid beta (1 to 42) (unknown origin) after 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50492186(CHEMBL2397722)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]IMPY from amyloid beta (1 to 42) (unknown origin) after 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50492182(CHEMBL2397724)
Affinity DataKi:  80nMAssay Description:Displacement of [125I]IMPY from amyloid beta (1 to 42) (unknown origin) after 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50492184(CHEMBL2397723)
Affinity DataKi:  117nMAssay Description:Displacement of [125I]IMPY from amyloid beta (1 to 42) (unknown origin) after 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50492181(CHEMBL2397725)
Affinity DataKi:  1.03E+3nMAssay Description:Displacement of [125I]IMPY from amyloid beta (1 to 42) (unknown origin) after 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50492185(CHEMBL2397726)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125I]IMPY from amyloid beta (1 to 42) (unknown origin) after 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed